SCHEMBL27612825

SCHEMBL27612825

COc1ccc(Nc2nc(NN3CCN(Cc4ccccc4)CC3)ncc2F)cc1OC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCL6 P41182 10/20 0.50
EGFR P00533 1/20 0.49
ITK Q08881 1/20 0.49
NCOR2 Q9Y618 1/20 0.48
ALDH1A1 P00352 2/20 0.47
LMNA P02545 2/20 0.47
POLB P06746 1/20 0.47
MAPT P10636 1/20 0.47
MAPK1 P28482 1/20 0.47
HTT P42858 1/20 0.47
ACHE P22303 1/20 0.47
BACE1 P56817 1/20 0.47
JAK3 P52333 1/20 0.45
BTK Q06187 1/20 0.45
AURKA O14965 1/20 0.45
AURKB Q96GD4 1/20 0.45
MAPK8 P45983 1/20 0.45
MAPK9 P45984 1/20 0.45
AXL P30530 1/20 0.45
BRD4 O60885 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL657262 0.88 BCL6 (0.55) BCL6EGFRITKNCOR2ALDH1A1
SCHEMBL656063 0.76 EGFR (0.69) BCL6EGFRITKNCOR2AURKA
SCHEMBL27631624 0.75 BCL6 (0.49) BCL6EGFRITKNCOR2ALDH1A1
SCHEMBL655906 0.74 SYK (0.65) EGFRITKJAK3BTKAURKA
SCHEMBL653516 0.71 BCL6 (0.59) BCL6EGFRITKNCOR2ALDH1A1
SCHEMBL657143 0.70 SYK (0.78) BCL6EGFRITKNCOR2AURKA
SCHEMBL655720 0.70 SYK (0.76) EGFRITKAURKA
SCHEMBL656282 0.70 SYK (0.76) EGFRITKAURKA
SCHEMBL655513 0.70 SYK (0.78) BCL6EGFRITKNCOR2AURKA
SCHEMBL656233 0.70 SYK (0.60) BCL6EGFRITKNCOR2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1678321-A Methods of treating or preventing autoimmune diseases with 2, 4-pyrimidinediamine compounds RIGEL PHARMACEUTICALS INC (US) 2005-10-05 CN disclosed