SCHEMBL27612843

SCHEMBL27612843

C/C=C/c1ccc(-c2cnccn2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.49
CYP2C9 P11712 2/20 0.49
CYP19A1 P11511 1/20 0.49
CYP2C19 P33261 1/20 0.49
PIM2 Q9P1W9 2/20 0.42
RAB9A P51151 2/20 0.41
KMT2A Q03164 1/20 0.41
BRS3 P32247 1/20 0.39
PIK3CD O00329 1/20 0.38
PIK3CA P42336 1/20 0.38
PIK3CB P42338 1/20 0.38
PI4KA P42356 1/20 0.38
PIK3CG P48736 1/20 0.38
PI4KB Q9UBF8 1/20 0.38
DHODH Q02127 1/20 0.38
TSHR P16473 3/20 0.37
CYP3A4 P08684 2/20 0.37
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.37
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6229775 0.82 CYP2D6 (0.45) CYP2D6CYP2C9CYP19A1CYP2C19PIM2
SCHEMBL6878325 0.81 CYP2D6 (0.49) CYP2D6CYP2C9CYP19A1CYP2C19PIM2
SCHEMBL6878319 0.81 CYP2D6 (0.49) CYP2D6CYP2C9CYP19A1CYP2C19PIM2
SCHEMBL11541937 0.80 CYP2D6 (0.60) CYP2D6CYP2C9CYP19A1CYP2C19PIM2
SCHEMBL6227552 0.79 PIM2 (0.43) CYP2D6CYP2C9CYP19A1CYP2C19PIM2
SCHEMBL6227545 0.79 PIM2 (0.43) CYP2D6CYP2C9CYP19A1CYP2C19PIM2
SCHEMBL6230889 0.78 CYP2D6 (0.45) CYP2D6CYP2C9CYP19A1CYP2C19PIM2
SCHEMBL6230887 0.78 CYP2D6 (0.45) CYP2D6CYP2C9CYP19A1CYP2C19PIM2
SCHEMBL6750 0.78 KDM4E (0.53) CYP2D6CYP2C9CYP19A1CYP2C19PIM2
SCHEMBL6276330 0.78 CYP2D6 (0.47) CYP2D6CYP2C9CYP19A1CYP2C19PIM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1585775-A 6-O-acyl ketolide derivatives of erythromycine useful as antibacterials ORTHO MCNEIL PHARM INC (US) 2005-02-23 CN disclosed