SCHEMBL27615016

SCHEMBL27615016

[CH2]CCNc1ncc(C(=O)c2ccccc2CC)s1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 9/20 0.44
MAPK13 O15264 8/20 0.44
MAPK12 P53778 8/20 0.44
MAPK11 Q15759 8/20 0.44
NPC1 O15118 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
RAB9A P51151 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6876510 0.86 MAPK14 (0.47) MAPK14MAPK13MAPK12MAPK11NPC1
SCHEMBL5564247 0.86 MAPK14 (0.43) MAPK14MAPK13MAPK12MAPK11NPC1
SCHEMBL5564238 0.86 MAPK14 (0.46) MAPK14MAPK13MAPK12MAPK11NPC1
SCHEMBL27596211 0.84 MAPK14 (0.64) MAPK14MAPK13MAPK12MAPK11NPC1
SCHEMBL5568870 0.82 POLB (0.44) MAPK14MAPK13MAPK12MAPK11NPC1
SCHEMBL27596159 0.82 MAPK13 (0.44) MAPK14MAPK13MAPK12MAPK11
SCHEMBL5565186 0.81 NPC1 (0.46) MAPK14MAPK13MAPK12MAPK11NPC1
SCHEMBL6879014 0.81 NPC1 (0.63) MAPK14MAPK13MAPK12MAPK11NPC1
SCHEMBL5564741 0.80 MAPK14 (0.45) MAPK14MAPK13MAPK12MAPK11NPC1
SCHEMBL5569153 0.80 MAPK13 (0.44) MAPK14MAPK13MAPK12MAPK11NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100363362-C Thiazole derivatives as NPY receptor antagonists HOFFMANN LA ROCHE (CH) 2008-01-23 CN disclosed
CN-1639158-A Thiazole derivatives as NPY receptor antagonists HOFFMANN LA ROCHE (CH) 2005-07-13 CN disclosed