SCHEMBL27624947

SCHEMBL27624947

Cc1ccc2c(c1)c(Sc1ccccc1CN)c(C)n2CC(=O)O

nearest known ligand 0.73

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 19/20 0.73
AKR1B1 P15121 8/20 0.73
CYP2C9 P11712 2/20 0.60
SLC6A2 P23975 1/20 0.45
SLC6A4 P31645 1/20 0.45
SLC6A3 Q01959 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3009395 0.91 PTGDR2 (0.76) PTGDR2AKR1B1CYP2C9
SCHEMBL1406036 0.86 PTGDR2 (0.79) PTGDR2AKR1B1CYP2C9SLC6A4
SCHEMBL28755766 0.86 PTGDR2 (0.69) PTGDR2AKR1B1CYP2C9
SCHEMBL1406169 0.84 PTGDR2 (0.76) PTGDR2AKR1B1CYP2C9
SCHEMBL1406026 0.84 PTGDR2 (1.00) PTGDR2AKR1B1CYP2C9
SCHEMBL1406010 0.83 PTGDR2 (0.73) PTGDR2AKR1B1CYP2C9
SCHEMBL5361236 0.82 PTGDR2 (0.82) PTGDR2AKR1B1CYP2C9
SCHEMBL1406116 0.77 PTGDR2 (0.79) PTGDR2AKR1B1CYP2C9
SCHEMBL1405915 0.77 PTGDR2 (0.65) PTGDR2AKR1B1CYP2C9SLC6A4
SCHEMBL1406070 0.77 PTGDR2 (0.74) PTGDR2AKR1B1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100404505-C Novel substituted indoles ASTRAZENECA AB (SE) 2008-07-23 CN claimed
CN-1671659-A Novel substituted indoles ASTRAZENECA AB (SE) 2005-09-21 CN claimed
CN-100404505-C Novel substituted indoles ASTRAZENECA AB (SE) 2008-07-23 CN disclosed
CN-1671659-A Novel substituted indoles ASTRAZENECA AB (SE) 2005-09-21 CN disclosed