SCHEMBL27626596

SCHEMBL27626596

CNC(=O)c1ccc(CCc2sc(NC(C)=O)nc2CCc2ccc(NC(=O)OC(C)(C)C)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 13/20 0.49
CYP17A1 P05093 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
NAMPT P43490 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
GLS O94925 1/20 0.41
LCK P06239 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4883904 0.91 AOC3 (0.48) AOC3CYP17A1HDAC1HDAC6RXFP1
SCHEMBL4867025 0.90 AOC3 (0.58) AOC3CYP17A1HDAC1HDAC6GLS
SCHEMBL28759633 0.88 AOC3 (0.46) AOC3CYP17A1HDAC1HDAC6GLS
SCHEMBL4866969 0.87 AOC3 (0.55) AOC3CYP17A1RXFP1GLS
SCHEMBL4874746 0.87 CYP17A1 (0.45) AOC3CYP17A1HDAC1HDAC6GLS
SCHEMBL4985325 0.86 AOC3 (0.52) AOC3SMN1; SMN2RXFP1
SCHEMBL27646813 0.86 AOC3 (0.46) AOC3CYP17A1HDAC1HDAC6RXFP1
SCHEMBL4878024 0.86 AOC3 (0.66) AOC3CYP17A1HDAC1HDAC6GLS
SCHEMBL4872960 0.86 AOC3 (0.55) AOC3CYP17A1SMN1; SMN2GLS
SCHEMBL14019606 0.84 AOC3 (0.53) AOC3SMN1; SMN2RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1794988-B Composition for treating vascular hyperpermeable disease SUCAMPO AG 2010-07-28 CN disclosed
CN-100491361-C Thiazole derivatives and their use as VAP-1 inhibitors FUJISAWA PHARMACEUTICAL CO (JP) 2009-05-27 CN disclosed
CN-1794988-A Method for treating vascular hyperpermeable disease SUCAMPO AG (CH) 2006-06-28 CN disclosed
CN-1761655-A Thiazole derivatives and their use as VAP-1 inhibitors FUJISAWA PHARMACEUTICAL CO (JP) 2006-04-19 CN disclosed