SCHEMBL2763353

SCHEMBL2763353

COc1ccc(Oc2ccncc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.59
SMN1; SMN2 Q16637 3/20 0.59
KDM4E B2RXH2 3/20 0.59
RAB9A P51151 3/20 0.59
CYP1A2 P05177 2/20 0.59
CYP2C9 P11712 2/20 0.59
CYP2C19 P33261 2/20 0.59
CYP3A4 P08684 1/20 0.59
CYP2D6 P10635 1/20 0.59
HPGD P15428 1/20 0.59
LTA4H P09960 2/20 0.58
MEN1 O00255 1/20 0.56
ALDH1A1 P00352 1/20 0.56
KMT2A Q03164 1/20 0.56
CA12 O43570 1/20 0.55
CA1 P00915 1/20 0.55
CA2 P00918 1/20 0.55
CA7 P43166 1/20 0.55
CA9 Q16790 1/20 0.55
CA14 Q9ULX7 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8213963 0.89 CYP1A2 (0.62) NPC1SMN1; SMN2KDM4ERAB9ACYP1A2
SCHEMBL61315 0.89
Ammonia Solution, Strong SCHEMBL28161848 0.87
SCHEMBL29452963 0.87
Hydrochloric Acid SCHEMBL27929151 0.87
Potassium SCHEMBL30601771 0.87
Hydroxyl Radical SCHEMBL28261927 0.87
Water SCHEMBL28135826 0.84 CYP1A2 (0.58) NPC1SMN1; SMN2KDM4ERAB9ACYP1A2
SCHEMBL11580995 0.84 CA1 (0.79) NPC1SMN1; SMN2KDM4ERAB9ACYP3A4
SCHEMBL166536 0.84 CA1 (0.79) NPC1SMN1; SMN2KDM4ERAB9ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100174089-A1 HETEROARYL ARYL ETHERS SALTIGO GMBH (DE) 2010-07-08 US claimed
EP-2179989-A2 Process for the preparation of heteroaryl - aryl ether Saltigo GmbH (DE) 2010-04-28 EP claimed
US-8592595-B2 Preparation of (N-heterocyclyl) aryl ethers SALTIGO GMBH (DE) 2013-11-26 US disclosed
US-20100174089-A1 HETEROARYL ARYL ETHERS SALTIGO GMBH (DE) 2010-07-08 US disclosed
US-20100152454-A1 PREPARATION OF (N-HETEROCYCLYL) ARYL ETHERS SALTIGO GMBH (DE) 2010-06-17 US disclosed
EP-2179989-A2 Process for the preparation of heteroaryl - aryl ether Saltigo GmbH (DE) 2010-04-28 EP disclosed
EP-2179988-A1 Producing (N-heterocyclic) aryl ethers Saltigo GmbH (DE) 2010-04-28 EP disclosed
US-4411904-A Diphenylpropanamines, compositions thereof and use thereof WARNER-LAMBERT COMPANY (US) 1983-10-25 US disclosed
US-4364954-A NEUROLEPTIC AGENT WARNER-LAMBERT COMPANY (US) 1982-12-21 US disclosed
US-4292321-A 1,3,8-Triazaspirodecane-4-ones, pharmaceutical compositions thereof and method of use thereof WARNER-LAMBERT COMPANY (US) 1981-09-29 US disclosed
US-4218456-A 1-(4-Fluorophenyl)-4-(1,2,3,6-tetrahydro-4-phenoxy-1-pyridinyl)-butanones WARNER-LAMBERT COMPANY (US) 1980-08-19 US disclosed