SCHEMBL27645010

SCHEMBL27645010

c1ccc(CC2CCN(c3ccc4ccccc4n3)CC2)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 6/20 0.64
HRH3 Q9Y5N1 4/20 0.57
ALDH1A1 P00352 4/20 0.54
KDM4E B2RXH2 3/20 0.54
HTR3E A5X5Y0 2/20 0.54
HTR3B O95264 2/20 0.54
CYP1A2 P05177 2/20 0.54
HTR3A P46098 2/20 0.54
HTR3D Q70Z44 2/20 0.54
HTR3C Q8WXA8 2/20 0.54
SLC6A4 P31645 2/20 0.54
TDP1 Q9NUW8 2/20 0.54
HTT P42858 2/20 0.54
USP2 O75604 1/20 0.54
ADRB1 P08588 1/20 0.54
CYP3A4 P08684 1/20 0.54
HTR1A P08908 1/20 0.54
HTR2C P28335 1/20 0.54
MAPK1 P28482 1/20 0.54
HTR7 P34969 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27644559 0.86 KDM4E (0.52) PDE10AHRH3ALDH1A1KDM4EHTR3E
SCHEMBL27645130 0.86 PDE10A (0.51) PDE10AHRH3ALDH1A1KDM4EHTR3E
SCHEMBL2596175 0.84 PDE10A (0.77) PDE10APDE2APDE1BPDE4DPDE11A
SCHEMBL27666226 0.82 PDE10A (0.54) PDE10AHRH3ALDH1A1KDM4EHTR3E
SCHEMBL2096494 0.81 ESR1 (0.54) PDE10AALDH1A1KDM4EHTTMAPK1
SCHEMBL237961 0.80 PDE10A (0.64) PDE10AHRH3ALDH1A1KDM4EHTR3E
SCHEMBL16454449 0.79 PDE10A (1.00) PDE10A
SCHEMBL16454485 0.79 PDE10A (1.00) PDE10A
SCHEMBL2596181 0.79 PDE10A (1.00) PDE10A
SCHEMBL2096492 0.79 TSHR (0.49) PDE10AALDH1A1KDM4EHTTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100497345-C 2, 3-dihydro-6-nitroimidazolo [2,1-b] oxazole compounds for the treatment of tuberculosis OTSUKA PHARMA CO LTD (JP) 2009-06-10 CN disclosed
CN-1878777-A 2,3-dihydro-6-nitroimidazo (2,1-b) oxazole compounds for the treatment of tuberculosis OTSUKA PHARMA CO LTD (JP) 2006-12-13 CN disclosed