SCHEMBL27646804

SCHEMBL27646804

CCOC(=O)NNc1nc(CCc2ccc(N)cc2)cs1

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 15/20 0.53
MAOB P27338 3/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
ALDH1A1 P00352 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4874642 0.88 AOC3 (0.61) AOC3MAOBHDAC1HDAC6ALDH1A1
SCHEMBL27626575 0.87 AOC3 (0.48) AOC3MAOBHDAC1HDAC6
SCHEMBL3406120 0.81 AOC3 (0.61) AOC3MAOB
SCHEMBL27646805 0.79 MAPK1 (0.46) ALDH1A1
SCHEMBL27646817 0.78 SMN1; SMN2 (0.55) ALDH1A1
SCHEMBL3934166 0.77 AOC3 (0.85) AOC3MAOB
SCHEMBL4873462 0.76 AOC3 (0.55) AOC3MAOBHDAC1HDAC6
SCHEMBL13679476 0.75 AOC3 (0.58) AOC3MAOB
Hydrochloric Acid SCHEMBL4876215 0.74 AOC3 (0.57) AOC3MAOB
SCHEMBL4876641 0.74 AOC3 (0.73) AOC3MAOBHDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100491361-C Thiazole derivatives and their use as VAP-1 inhibitors FUJISAWA PHARMACEUTICAL CO (JP) 2009-05-27 CN disclosed
CN-1761655-A Thiazole derivatives and their use as VAP-1 inhibitors FUJISAWA PHARMACEUTICAL CO (JP) 2006-04-19 CN disclosed