SCHEMBL27653232

SCHEMBL27653232

Cc1n[nH]c(-c2ccccc2)c1C(Cc1ccccc1)C(N)=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.49
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
MMP3 P08254 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
PTPN1 P18031 1/20 0.37
PPARG P37231 5/20 0.37
PPARA Q07869 5/20 0.37
BACE1 P56817 1/20 0.37
BACE2 Q9Y5Z0 1/20 0.37
CPA1 P15085 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36
MME P08473 1/20 0.36
ELANE P08246 1/20 0.36
ALPI P09923 1/20 0.36
PKM P14618 1/20 0.36
PTGS1 P23219 1/20 0.36
XIAP P98170 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27653231 0.75 DCAF1 (0.46) ALDH1A1RAB9A
SCHEMBL22897288 0.72 CAPN1 (0.54)
SCHEMBL20028370 0.72 CAPN1 (0.54)
SCHEMBL20148796 0.71 AKT2 (0.47) MEN1KMT2AALDH1A1RAB9A
SCHEMBL2109313 0.68 EPHX1 (0.68) EPHX1PPARGPPARACPA1ALDH1A1
SCHEMBL1516139 0.67 EPHX1 (1.00) EPHX1ALDH1A1ALPIPKMPTGS1
SCHEMBL28107950 0.67 EPHX1 (0.77) EPHX1MEN1KMT2APPARGPPARA
SCHEMBL14678497 0.67 EPHX1 (0.62) EPHX1MEN1KMT2AHDAC8PPARG
SCHEMBL13615358 0.67 CHEK1 (0.46) MEN1KMT2AALDH1A1RAB9A
SCHEMBL8620330 0.66 EPHX1 (0.96) EPHX1MEN1KMT2AALDH1A1ALPI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1802373-A Pyrazoloisoquinoline derivatives as kinase inhibitors AVENTIS PHARMA INC (US) 2006-07-12 CN disclosed