SCHEMBL27657151

SCHEMBL27657151

Cc1sc(-c2ccc(C(F)(F)F)cc2)nc1CCBr

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.46
ALDH1A1 P00352 1/20 0.46
GAA P10253 1/20 0.46
MAPT P10636 3/20 0.44
KDM4E B2RXH2 1/20 0.44
MEN1 O00255 1/20 0.44
HSP90AA1 P07900 1/20 0.44
CRHBP P24387 1/20 0.44
KMT2A Q03164 1/20 0.44
CRHR2 Q13324 1/20 0.44
CTSS P25774 1/20 0.44
MAOB P27338 1/20 0.42
PPARD Q03181 5/20 0.40
PPARG P37231 4/20 0.40
PPARA Q07869 4/20 0.40
FFAR1 O14842 3/20 0.40
SIRT2 Q8IXJ6 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
DCK P27707 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5017198 0.88 NPC1 (0.48) NPC1ALDH1A1GAAMAPTKDM4E
SCHEMBL4902987 0.86 MAOB (0.50) NPC1ALDH1A1GAAMAPTKDM4E
SCHEMBL968444 0.86 NPC1 (0.49) NPC1ALDH1A1GAAMAPTKDM4E
SCHEMBL18015833 0.84 MAPT (0.50) NPC1ALDH1A1GAAMAPTKDM4E
SCHEMBL4466375 0.83 NPC1 (0.47) NPC1ALDH1A1GAAMAPTKDM4E
SCHEMBL5102703 0.82 MAPT (0.52) NPC1ALDH1A1GAAMAPTKDM4E
SCHEMBL27670372 0.82 NPC1 (0.48) NPC1ALDH1A1GAAMAPTKDM4E
SCHEMBL20642197 0.82 NPC1 (0.48) NPC1ALDH1A1GAAMAPTKDM4E
SCHEMBL18014742 0.81 NPC1 (0.47) NPC1ALDH1A1GAAMAPTKDM4E
SCHEMBL27611734 0.81 MAPT (0.49) NPC1ALDH1A1GAAMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1816550-B Indolyl derivatives substituted with a thiazole ring and their use as PPAR modulators HOFFMANN LA ROCHE 2010-04-28 CN disclosed
CN-1816550-A Indolyl derivatives substituted with a thiazole ring and their use as ppar modulators HOFFMANN LA ROCHE (CH) 2006-08-09 CN disclosed