SCHEMBL27657166

SCHEMBL27657166

CC(C(=O)C(C)c1ccc(-c2ccnc(NC3CC(C)(C)NC(C)(C)C3)n2)s1)c1ccc(-c2ccnc(NC3CC(C)(C)NC(C)(C)C3)n2)s1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.38
CDK4 P11802 7/20 0.35
CCND1 P24385 7/20 0.35
CDK2 P24941 7/20 0.35
CDK1 P06493 6/20 0.35
CCNB1 P14635 6/20 0.35
CCNA2 P20248 6/20 0.35
CCNA1 P78396 6/20 0.35
CCND3 P30281 3/20 0.35
CDK6 Q00534 3/20 0.35
CCNE1 P24864 1/20 0.35
KMT2A Q03164 1/20 0.35
AURKA O14965 1/20 0.34
TTK P33981 1/20 0.34
AURKB Q96GD4 1/20 0.34
INCENP Q9NQS7 1/20 0.34
POLB P06746 1/20 0.34
MAPK8 P45983 3/20 0.34
MAPK9 P45984 3/20 0.34
AKT3 Q9Y243 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4484868 0.87 KCNH2 (0.37) KCNH2CDK4CCND1CDK2CDK1
SCHEMBL4489828 0.86 CDK1 (0.41) KCNH2CDK4CCND1CDK2CDK1
SCHEMBL27842465 0.86 KMT2A (0.39) KCNH2CDK4CCND1CDK2CDK1
SCHEMBL27657167 0.86 KCNH2 (0.36) KCNH2CDK4CCND1CDK2CDK1
SCHEMBL3478664 0.84 CDK1 (0.40) KCNH2CDK4CCND1CDK2CDK1
SCHEMBL27842563 0.83 KCNH2 (0.38) KCNH2CDK2CCNA2AURKATTK
SCHEMBL4491124 0.82 AKT3 (0.42) KCNH2CDK4CCND1CDK2CDK1
SCHEMBL3470259 0.82 AKT3 (0.42) KCNH2CDK4CCND1CDK2CDK1
SCHEMBL3472051 0.81 IKBKB (0.41) KCNH2CDK2CCNA2MAPK8MAPK9
SCHEMBL3476590 0.80 AKT3 (0.41) KCNH2CDK4CCND1CDK2CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102267988-A 2-aminopyrimidine derivatives and their medical use NOVARTIS LTD 2011-12-07 CN disclosed
CN-1802357-A 2-aminopyrimidine derivatives and their medical use NOVARTIS AG (CH) 2006-07-12 CN disclosed