SCHEMBL27657306

SCHEMBL27657306

NC(=O)N(c1ccc(-c2cccc3[nH]nc(N)c23)c(F)c1)c1ccc(F)c(C(F)(F)F)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 14/20 0.58
KIT P10721 8/20 0.51
FLT3 P36888 8/20 0.51
CSF1R P07333 7/20 0.51
FLT1 P17948 7/20 0.51
LCK P06239 6/20 0.51
LYN P07948 6/20 0.51
SRC P12931 6/20 0.51
FLT4 P35916 6/20 0.51
BLK P51451 6/20 0.51
FYN P06241 4/20 0.48
ABL1 P00519 9/20 0.43
BCR P11274 6/20 0.43
CDK19 Q9BWU1 2/20 0.42
NTRK1 P04629 2/20 0.41
RET P07949 2/20 0.41
MET P08581 2/20 0.41
PDGFRB P09619 2/20 0.41
FGFR1 P11362 2/20 0.41
PRKACA P17612 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27657344 0.91 KDR (0.69) KDRKITFLT3CSF1RFLT1
SCHEMBL27657342 0.86 KDR (0.57) KDRKITFLT3CSF1RFLT1
SCHEMBL13372697 0.86 KDR (0.65) KDRKITFLT3CSF1RFLT1
SCHEMBL28760140 0.86 KDR (0.62) KDRKITFLT3CSF1RFLT1
SCHEMBL27636479 0.85 KDR (0.66) KDRKITFLT3CSF1RFLT1
SCHEMBL27657464 0.85 KDR (0.55) KDRKITFLT3CSF1RFLT1
SCHEMBL3422842 0.84 KDR (0.56) KDRKITFLT3CSF1RFLT1
SCHEMBL27636383 0.83 KDR (0.53) KDRKITFLT3CSF1RFLT1
SCHEMBL27657395 0.81 KDR (0.51) KDRKITFLT3CSF1RFLT1
SCHEMBL27657361 0.80 KDR (0.62) KDRKITFLT3CSF1RFLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1826324-B indazole, Benzisoxazole and benzisothiazole kinase inhibitors ABBOTT LABORATORIES (US) 2011-12-07 CN claimed
CN-1826324-A Indazole, benzisoxazole and benzisothiazole kinase inhibitors ABBOTT LAB (US) 2006-08-30 CN claimed
CN-102417487-A Indazole, benzisoxazole and benzisothiazole kinase inhibitors ABBOTT LAB 2012-04-18 CN disclosed
CN-1826324-B indazole, Benzisoxazole and benzisothiazole kinase inhibitors ABBOTT LABORATORIES (US) 2011-12-07 CN disclosed
CN-101827584-A Solid dispersion product of N-aryl ureido drugs ABBOTT GMBH & CO KG 2010-09-08 CN disclosed
CN-1826324-A Indazole, benzisoxazole and benzisothiazole kinase inhibitors ABBOTT LAB (US) 2006-08-30 CN disclosed