SCHEMBL27657404

SCHEMBL27657404

Nc1ncccc1-c1cc[c]s1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.42
MKNK1 Q9BUB5 2/20 0.39
MKNK2 Q9HBH9 2/20 0.39
NOS3 P29474 2/20 0.38
NOS1 P29475 2/20 0.38
NOS2 P35228 2/20 0.38
CDK1 P06493 1/20 0.37
CDK2 P24941 1/20 0.37
PDGFRB P09619 3/20 0.34
KDR P35968 3/20 0.34
NAPRT Q6XQN6 1/20 0.34
LTA4H P09960 1/20 0.34
MAPK14 Q16539 1/20 0.34
AKT1 P31749 3/20 0.33
PI4KA P42356 1/20 0.33
PI4K2B Q8TCG2 1/20 0.33
PI4K2A Q9BTU6 1/20 0.33
PI4KB Q9UBF8 1/20 0.33
AKT2 P31751 1/20 0.33
TGFBR1 P36897 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5917511 0.79 NPC1 (0.36) NPC1RAB9ASMN1; SMN2S100A4MEN1
SCHEMBL27657456 0.78 CA12 (0.43) MAPT
SCHEMBL3539250 0.76 KDM4E (0.48) CDK2HTTNPC1RAB9ASMN1; SMN2
SCHEMBL10062975 0.73 MAP4K4 (0.59) MAP4K4MKNK1MKNK2NOS3NOS1
SCHEMBL3596326 0.72 CYP2A6 (0.35) NOS3NOS1NOS2PI4KAPI4K2B
SCHEMBL30968134 0.71 MAP4K4 (0.57) MAP4K4MKNK1MKNK2NOS3NOS1
SCHEMBL27401952 0.70 NPC1 (0.47) MAP4K4MKNK1MKNK2NOS3NOS1
SCHEMBL27657405 0.69 CYP1A2 (0.44) MAPK14TGFBR1NPC1RAB9ASMN1; SMN2
SCHEMBL295633 0.68 KDM4E (0.57) HTTNPC1RAB9ASMN1; SMN2LMNA
SCHEMBL3845483 0.68 MAP4K4 (0.55) MAP4K4MKNK1MKNK2NOS3NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1829721-A Spiro '1-azabicyclo' 2.2.2! octan-3,5'-oxazolidin - 2'-one! derivatives with affinity to the alpha7 nicotinic acetylcholine receptor ASTRAZENECA AB (SE) 2006-09-06 CN claimed
CN-1829721-A Spiro '1-azabicyclo' 2.2.2! octan-3,5'-oxazolidin - 2'-one! derivatives with affinity to the alpha7 nicotinic acetylcholine receptor ASTRAZENECA AB (SE) 2006-09-06 CN disclosed