SCHEMBL27675752

SCHEMBL27675752

NC(=O)c1ccccc1-c1[nH]c2ccsc2c1Sc1cccc(Br)c1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 2/20 0.36
MAPK8 P45983 1/20 0.36
SIRT1 Q96EB6 2/20 0.34
TYMS P04818 2/20 0.34
PARP1 P09874 6/20 0.32
BCAT2 O15382 1/20 0.32
KDR P35968 1/20 0.31
AURKA O14965 1/20 0.31
RPS6KB1 P23443 1/20 0.31
NCOA1 Q15788 1/20 0.31
NCOA3 Q9Y6Q9 1/20 0.31
PIM1 P11309 1/20 0.31
CSNK2B P67870 1/20 0.31
CSNK2A1 P68400 1/20 0.31
PIM2 Q9P1W9 1/20 0.31
ALDH1A1 P00352 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27694235 0.89 KDR (0.37) CDC7MAPK8SIRT1TYMSPARP1
SCHEMBL27694282 0.86 EDNRA (0.44) CDC7MAPK8PARP1
SCHEMBL27675744 0.85 CDC7 (0.37) CDC7MAPK8SIRT1TYMSPARP1
SCHEMBL27694283 0.84 BRD4 (0.34) CDC7MAPK8SIRT1PARP1BCAT2
SCHEMBL28763133 0.84 CHEK1 (0.33) PARP1BCAT2PIM1CSNK2BCSNK2A1
SCHEMBL27675745 0.83 BCL2L1 (0.36) SIRT1PARP1BCAT2PIM1CSNK2B
SCHEMBL27675746 0.83 CDC7 (0.39) CDC7SIRT1PARP1BCAT2RPS6KB1
SCHEMBL3175305 0.82 TYMS (0.37) CDC7MAPK8TYMSPARP1KDR
SCHEMBL28763131 0.80 PDE7A (0.37) CDC7SIRT1PARP1BCAT2ALDH1A1
SCHEMBL27694287 0.79 NPC1 (0.41) CDC7MAPK8SIRT1PARP1BCAT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100562521-C Substituted thienopyrrole carboxylic acid amides, pyrrolothiazole carboxylic acid amides, and related analogs as inhibitors of casein kinase ie AVENTIS PHARMA INC (US) 2009-11-25 CN disclosed
CN-101001861-A Substituted thienopyrrole carboxylic acid amides, pyrrolothiazole carboxylic acid amides, and related analogs as inhibitors of casein kinase i epsilon AVENTIS PHARMA INC (US) 2007-07-18 CN disclosed