SCHEMBL27675982

SCHEMBL27675982

N[C@@H]1Cc2cccnc2NC1C=O

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.35
IDH1 O75874 8/20 0.34
TRIM24 O15164 1/20 0.31
TRIM33 Q9UPN9 1/20 0.31
TNKS2 Q9H2K2 1/20 0.31
CYP1A2 P05177 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27676062 1.00 GSK3B (0.35) GSK3BIDH1TRIM24TRIM33TNKS2
SCHEMBL27676121 1.00 GSK3B (0.35) GSK3BIDH1TRIM24TRIM33TNKS2
SCHEMBL27600814 0.79 GSK3B (0.32) GSK3B
Hydrochloric Acid SCHEMBL27619412 0.78 GSK3B (0.31) GSK3B
SCHEMBL27458227 0.78 GSK3B (0.35) GSK3BIDH1TRIM24TRIM33TNKS2
SCHEMBL24096704 0.76 IDH1 (0.36) GSK3BIDH1
SCHEMBL27299860 0.76 GAA (0.46)
SCHEMBL4183810 0.75 GSK3B (0.34) GSK3BIDH1TNKS2
Hydrochloric Acid SCHEMBL27619269 0.74 GAA (0.45)
SCHEMBL27798345 0.72 CD44 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101001841-A Tetrahydroquinolones and aza-analogues thereof useful as DPP-IV inhibitors for the treatment of diabetes ASTRAZENECA AB (SE) 2007-07-18 CN disclosed