SCHEMBL2767668

SCHEMBL2767668

C[C@H]1CN(Cc2ccc(N(C)C(=O)C3CCN(Cc4cccc(F)c4)CC3)cc2)CCN1C(=O)O

nearest known ligand 0.72

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MLNR O43193 5/20 0.72
CCR5 P51681 3/20 0.51
ALDH1A1 P00352 1/20 0.48
ACHE P22303 1/20 0.44
CHRM4 P08173 1/20 0.44
F10 P00742 1/20 0.44
CCR1 P32246 1/20 0.44
SIGMAR1 Q99720 2/20 0.44
KMT2A Q03164 1/20 0.44
DRD2 P14416 2/20 0.44
DRD4 P21917 2/20 0.44
CACNA1G O43497 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2767709 0.91 MLNR (0.69) MLNRCCR5ALDH1A1CCR1CACNA1G
SCHEMBL2766379 0.89 MLNR (0.58) MLNRCCR5ALDH1A1CCR1SIGMAR1
SCHEMBL13404693 0.88 MLNR (0.66) MLNRCCR5ALDH1A1ACHECHRM4
SCHEMBL2766816 0.88 MLNR (0.57) MLNRCCR5ALDH1A1KMT2A
SCHEMBL3556504 0.87 MLNR (0.75) MLNRCCR5CHRM4
SCHEMBL2767269 0.84 MLNR (1.00) MLNR
SCHEMBL2766459 0.84 MLNR (0.60) MLNRCCR5CHRM4CCR1
SCHEMBL3558154 0.83 MLNR (0.72) MLNRCCR5ALDH1A1CHRM4
SCHEMBL15152692 0.81 MLNR (0.51) MLNRCCR5ALDH1A1CCR1DRD4
SCHEMBL15152914 0.81 MLNR (0.56) MLNRCCR5CCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2041093-B1 PIPERAZINYL DERIVATIVES USEFUL IN THE TREATMENT OF GPR38 RECEPTOR MEDIATED DISEASES GLAXO GROUP LTD (GB) 2010-04-21 EP disclosed