SCHEMBL27680332

SCHEMBL27680332

NCc1cccc(Nc2ncnc3ccc(N)cc23)c1

nearest known ligand 0.68

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
EGFR P00533 18/20 0.68
ERBB2 P04626 3/20 0.68
AHR P35869 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29690398 0.82 EGFR (1.00) EGFRERBB2AHR
SCHEMBL30513 0.82 EGFR (1.00) EGFRERBB2AHR
SCHEMBL159209 0.81 EGFR (1.00) EGFRERBB2
SCHEMBL31060998 0.81 EGFR (1.00) EGFRERBB2
SCHEMBL29350058 0.81 EGFR (1.00) EGFRERBB2
SCHEMBL31060510 0.81 EGFR (1.00) EGFRERBB2
SCHEMBL4586872 0.81 EGFR (0.80) EGFRERBB2AHR
SCHEMBL14578431 0.81 EGFR (0.72) EGFRERBB2AHR
SCHEMBL1262804 0.81 EGFR (1.00) EGFRERBB2
SCHEMBL10108264 0.81 EGFR (0.72) EGFRERBB2AHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 55 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109963871-A Multivalence and multi-epitope Antibody and application method with agonist activity 豪夫迈·罗氏有限公司 2019-07-02 CN disclosed
CN-109312407-A Diagnostic and therapeutic method for cancer 豪夫迈·罗氏有限公司 2019-02-05 CN disclosed
CN-109053891-A A kind of anti-PD-L1 antibody and its preparation method and application 苏州泓迅生物科技股份有限公司 2018-12-21 CN disclosed
CN-108697713-A Methods for making tricyclic PI3K inhibitor compounds and methods of treating cancer therewith 基因泰克公司 2018-10-23 CN disclosed
CN-108026110-A Fused tricyclic compounds as kinases inhibitor 国家公共部门基金会卡洛斯三世国家癌症研究中心(F.S.P.CNIO) 2018-05-11 CN disclosed
CN-107912040-A Pyrrolidine Amide Compounds As Histone Demethylase Inhibitors 基因泰克公司 2018-04-13 CN disclosed
CN-107531690-A The amines of 4,5,6,7 tetrahydrochysene 1H pyrazolos [4,3 c] pyridine 3 as CBP and/or EP300 inhibitor 基因泰克公司 2018-01-02 CN disclosed
CN-107406414-A (piperidin-3-yl) (naphthalen-2-yl) methanone derivatives and related compounds as inhibitors of histone demethylase KDM2B for the treatment of cancer 基因泰克公司 2017-11-28 CN disclosed
CN-107406418-A 4,5 glyoxalidine derivatives and its purposes as histone demethylase (KDM2B) inhibitor 基因泰克公司 2017-11-28 CN disclosed
CN-107406429-A Pyridazinone derivative and its purposes in treating cancer 基因泰克公司 2017-11-28 CN disclosed
CN-101023100-B Her2 antibody composition GENENTECH INC 2012-08-29 CN disclosed
CN-102612374-A A method of promoting dendritic spine density HOFFMANN LA ROCHE 2012-07-25 CN disclosed
CN-102356092-A Bispecific anti-her antibodies GENENTECH INC 2012-02-15 CN disclosed
CN-102216331-A Method of treatment HOFFMANN LA ROCHE 2011-10-12 CN disclosed
CN-102124336-A Method for screening for compounds that inhibit neurodegeneration GENENTECH INC 2011-07-13 CN disclosed
CN-102014913-A Combination therapy with C-MET and EGFR antagonists GENENTECH INC 2011-04-13 CN disclosed
CN-101981056-A Composition comprising antibody that binds to domain II of HER2 and acidic variants thereof GENENTECH INC 2011-02-23 CN disclosed
CN-101616934-A Suppress DR6 antibody and the purposes in treatment neuroscience illness thereof of DR6 in conjunction with APP GENENTECH INC 2009-12-30 CN disclosed
CN-101180072-A Methods of using death receptor agonists and egfr inhibitors GENENTECH INC (US) 2008-05-14 CN disclosed
CN-101023100-A HER2 antibody composition GENENTECH INC 2007-08-22 CN disclosed