SCHEMBL27680916

SCHEMBL27680916

O=C(CCc1cccnc1)Nc1ccc(-c2nc(-c3cccc(CO)c3)ncc2C2CNCCO2)cc1

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 2/20 0.39
HPGDS O60760 1/20 0.39
PSMB8 P28062 1/20 0.38
SLC6A3 Q01959 1/20 0.38
KCNH2 Q12809 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38
CDK8 P49336 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27680915 0.86 NAMPT (0.40) NAMPTHPGDSPSMB8SLC6A3KCNH2
SCHEMBL27705032 0.78 ABL1 (0.43) SLC6A3KCNH2TAAR1
SCHEMBL27680900 0.78 ABL1 (0.43) SLC6A3KCNH2TAAR1
SCHEMBL27680902 0.75 CYP1A2 (0.40)
SCHEMBL27685979 0.75 CYP1A2 (0.40)
SCHEMBL27685994 0.72 PIP5K1C (0.42) SLC6A3KCNH2TAAR1
SCHEMBL4936580 0.71 PIK3CA (0.55)
SCHEMBL28764798 0.70 TAAR1 (0.42) SLC6A3KCNH2TAAR1
SCHEMBL27700077 0.69 MOK (0.44) TAAR1
SCHEMBL27700089 0.69 PIK3CA (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101010317-A 2, 4,6-trisubstituted pyrimidines as phosphotidylinositol (pi) 3-kinase inhibitors and their use in the treatment of cancer ASTRAZENECA AB (SE) 2007-08-01 CN disclosed