SCHEMBL27681237

SCHEMBL27681237

CC(F)C(=O)Nc1cc(-n2cccn2)nc(-c2ccco2)n1

nearest known ligand 0.76

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 17/20 0.76
ADORA1 P30542 16/20 0.76
ADORA3 P0DMS8 7/20 0.63
ADORA2B P29275 5/20 0.63
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5017911 0.92 ADORA2A (0.79) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL5017677 0.86 ADORA2A (1.00) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL5017746 0.86 ADORA2A (0.76) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL5016065 0.85 ADORA2A (0.82) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL27661824 0.85 ADORA2A (0.55) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL5016215 0.85 ADORA2A (0.76) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL5016198 0.85 ADORA2A (0.68) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL5612886 0.84 ADORA2A (0.80) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL5022598 0.84 ADORA2A (0.79) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL5017646 0.84 ADORA2A (0.80) ADORA2AADORA1ADORA3ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1953975-A 2, 6 bisheteroaryl-4-aminopyrimidines as adenosine receptor antagonists ALMIRALL PRODESFARMA AG (CH) 2007-04-25 CN claimed
CN-1953975-A 2, 6 bisheteroaryl-4-aminopyrimidines as adenosine receptor antagonists ALMIRALL PRODESFARMA AG (CH) 2007-04-25 CN disclosed