SCHEMBL27683093

SCHEMBL27683093

C/C(C(=O)O)=C(\C(=O)O)C(F)(F)F.CNC(CC(C)C)C(=O)N1CCC(N(C2CC2)S(=O)(=O)c2ccccc2)CC1

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 17/20 0.40
NR1I2 O75469 6/20 0.40
CCR1 P32246 1/20 0.39
CYP3A4 P08684 1/20 0.37
F2 P00734 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4282396 0.84 CACNA1B (0.51) CACNA1BNR1I2CYP3A4
SCHEMBL4277906 0.84 CACNA1B (0.51) CACNA1BNR1I2CYP3A4
SCHEMBL4280157 0.82 CACNA1B (0.60) CACNA1BNR1I2CYP3A4
SCHEMBL4278747 0.82 CACNA1B (0.60) CACNA1BNR1I2CYP3A4
SCHEMBL4277799 0.82 CACNA1B (0.60) CACNA1BNR1I2CYP3A4
SCHEMBL4285271 0.80 HTR2A (0.45) CACNA1BNR1I2CCR1CYP3A4F2
SCHEMBL4277967 0.80 HTR2A (0.45) CACNA1BNR1I2CCR1CYP3A4F2
SCHEMBL4277963 0.80 CACNA1B (0.48) CACNA1BNR1I2CYP3A4
SCHEMBL4282559 0.80 CACNA1B (0.42) CACNA1BNR1I2CCR1F2
SCHEMBL4282565 0.80 CACNA1B (0.42) CACNA1BNR1I2CCR1F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101044116-A 4-phenylsulfonamidopiperidines as calcium channel blockers EURO CELTIQUE SA (LU) 2007-09-26 CN disclosed