SCHEMBL27698705

SCHEMBL27698705

COCCOc1cc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2cc1NC(=O)C(C)N

nearest known ligand 0.79

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EGFR P00533 20/20 0.79
ERBB2 P04626 8/20 0.69
ERBB4 Q15303 3/20 0.69
GAK O14976 1/20 0.64
HDAC3 O15379 1/20 0.61
HDAC4 P56524 1/20 0.61
HDAC1 Q13547 1/20 0.61
HDAC7 Q8WUI4 1/20 0.61
HDAC2 Q92769 1/20 0.61
HDAC10 Q969S8 1/20 0.61
HDAC11 Q96DB2 1/20 0.61
HDAC8 Q9BY41 1/20 0.61
HDAC6 Q9UBN7 1/20 0.61
HDAC9 Q9UKV0 1/20 0.61
HDAC5 Q9UQL6 1/20 0.61
JAK3 P52333 2/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2248340 1.00 EGFR (0.79) EGFRERBB2ERBB4GAKHDAC3
SCHEMBL2249186 0.90 EGFR (0.81) EGFRERBB2ERBB4GAKHDAC3
SCHEMBL2248342 0.89 EGFR (0.80) EGFRERBB2ERBB4GAKHDAC3
SCHEMBL2249387 0.89 EGFR (0.85) EGFRERBB2ERBB4GAKHDAC2
SCHEMBL2249385 0.89 EGFR (0.85) EGFRERBB2ERBB4GAKHDAC2
SCHEMBL2248427 0.86 EGFR (0.72) EGFRERBB2ERBB4HDAC3HDAC4
SCHEMBL2255059 0.84 EGFR (0.87) EGFRERBB2ERBB4GAKHDAC3
SCHEMBL4865102 0.84 EGFR (0.75) EGFRERBB2ERBB4GAKHDAC3
SCHEMBL20412221 0.84 EGFR (0.82) EGFRERBB2ERBB4GAKHDAC3
SCHEMBL2249817 0.84 EGFR (0.78) EGFRERBB2ERBB4GAKHDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101094840-B Quinazoline derivatives for inhibiting the growth of cancer cells and methods for preparing the same HANMI PHARM IND CO LTD 2012-10-31 CN disclosed
CN-101094840-A Quinazoline derivatives for inhibiting the growth of cancer cells and methods for preparing the same HANMI PHARM IND CO LTD (KR) 2007-12-26 CN disclosed