SCHEMBL27700652

SCHEMBL27700652

O=[N+]([O-])c1cccc(-c2nc(Cl)nc3ccccc23)c1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.71
OPRK1 P41145 1/20 0.71
ALDH1A1 P00352 6/20 0.57
MAPT P10636 4/20 0.57
THRB P10828 1/20 0.57
TDP1 Q9NUW8 1/20 0.57
MEN1 O00255 3/20 0.56
GUSB P08236 1/20 0.56
ELANE P08246 1/20 0.56
POLB P06746 3/20 0.54
GAA P10253 2/20 0.54
LMNA P02545 1/20 0.54
HPGD P15428 1/20 0.54
ABCG2 Q9UNQ0 4/20 0.53
CFTR P13569 2/20 0.52
NPC1 O15118 1/20 0.51
RAB9A P51151 1/20 0.51
KDM4E B2RXH2 2/20 0.50
CYP1A2 P05177 1/20 0.50
PDE5A O76074 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1878028 0.87 KMT2A (0.72) KMT2AOPRK1ALDH1A1MAPTTHRB
SCHEMBL11706982 0.83 KMT2A (1.00) KMT2AOPRK1ALDH1A1MAPTMEN1
SCHEMBL12580134 0.83 KMT2A (0.59) KMT2AOPRK1ALDH1A1MAPTTHRB
SCHEMBL1941459 0.80 KMT2A (0.59) KMT2AOPRK1ALDH1A1MAPTMEN1
SCHEMBL27635805 0.80 NPC1 (0.62) KMT2AOPRK1ALDH1A1MAPTTHRB
SCHEMBL15538738 0.79 KDM4E (0.61) KMT2AOPRK1ALDH1A1MAPTTHRB
SCHEMBL28060242 0.79 NPC1 (0.66) KMT2AALDH1A1MAPTTHRBTDP1
SCHEMBL874141 0.78 POLB (0.67) KMT2AALDH1A1MAPTTHRBTDP1
SCHEMBL19293871 0.78 KDM4E (0.59) KMT2AOPRK1ALDH1A1MAPTTHRB
SCHEMBL16475867 0.78 KDM4E (0.64) KMT2AOPRK1ALDH1A1MAPTTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101180278-B 2-amino-4-phenylquinazoline derivates and their use as HSP90 modulators MERCK PATENT GMBH 2011-05-04 CN disclosed
CN-101180278-A 2-amino-4-phenylquinazoline derivates and their use as HSP90 modulators MERCK PATENT GMBH (DE) 2008-05-14 CN disclosed