SCHEMBL27700855

SCHEMBL27700855

CC(C)(C)OC(=O)N(CC(=O)Oc1ccc(-c2nn(C3CCCC3)c3c(F)cccc23)cc1)C(=O)CN

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.51
BTK Q06187 11/20 0.39
CMKLR1 Q99788 4/20 0.36
EGFR P00533 3/20 0.35
PTGDR2 Q9Y5Y4 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4027938 0.82 ESR1 (0.61) ESR1BTKCMKLR1EGFR
SCHEMBL4031427 0.81 ESR1 (0.65) ESR1BTKCMKLR1EGFR
SCHEMBL4030883 0.79 ESR1 (0.68) ESR1BTKCMKLR1EGFR
SCHEMBL4029342 0.78 ESR1 (0.69) ESR1BTKCMKLR1EGFR
SCHEMBL4027998 0.77 ESR1 (0.49) ESR1BTKCMKLR1
SCHEMBL5414144 0.76 ESR1 (0.52) ESR1BTKCMKLR1EGFR
SCHEMBL4028037 0.75 ESR1 (0.61) ESR1BTKCMKLR1EGFR
SCHEMBL27573477 0.73 ESR1 (0.45) ESR1BTK
SCHEMBL27573478 0.73 ESR1 (0.45) ESR1BTK
SCHEMBL4031188 0.73 ESR1 (0.72) ESR1BTKCMKLR1EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101054364-A Substituted 4-(indazol-3-yl)phenols as estrogen receptor (ER) ligands and their use in the treatmentof inflammarory diseases WYETH CORP (US) 2007-10-17 CN claimed