SCHEMBL27701710

SCHEMBL27701710

Cc1nc2ccc(Br)c(C)n2c1NC(C)C(=O)NO

nearest known ligand 0.32

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.32
HDAC1 Q13547 1/20 0.30
XIAP P98170 1/20 0.30
BIRC2 Q13490 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27701661 0.85 HDAC1 (0.33) HDAC1
SCHEMBL27722207 0.85 CHRNA1 (0.31) HDAC1
SCHEMBL27701753 0.84 CHRM1 (0.33) HDAC1
SCHEMBL27701650 0.75 GAA (0.32) GAAHDAC1
SCHEMBL27722225 0.68 HDAC1 (0.34) HDAC1
SCHEMBL27722260 0.65 HDAC1 (0.36) GAAHDAC1
SCHEMBL27722199 0.64 KDM4E (0.39) GAAHDAC1
SCHEMBL27722263 0.64 HDAC1 (0.35) HDAC1
SCHEMBL27722344 0.63 NR1H4 (0.30)
SCHEMBL27701721 0.63 GRIN1 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101163703-B Imidazo [1,2-A ] pyridine derivatives as Peptide Deformylase (PDF) inhibitors NOVARTIS AG 2010-12-15 CN disclosed
CN-101163703-A Imidazo [1, 2-A ] pyridine derivatives as Peptide Deformylase (PDF) inhibitors NOVARTIS AG (CH) 2008-04-16 CN disclosed