SCHEMBL2770352

SCHEMBL2770352

Cc1cc(OCc2c(C(C)C)cnn2-c2c(Cl)cccc2Cl)ccc1-c1ccc(C(=O)O)cn1

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 17/20 0.61
MRGPRX4 Q96LA9 1/20 0.40
VDR P11473 2/20 0.39
GCK P35557 1/20 0.37
LIFR P42702 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2770495 0.91 NR1H4 (0.67) NR1H4MRGPRX4VDRLIFR
SCHEMBL2771697 0.90 NR1H4 (0.63) NR1H4MRGPRX4VDR
SCHEMBL2772894 0.87 NR1H4 (0.67) NR1H4MRGPRX4LIFR
SCHEMBL2771465 0.85 NR1H4 (0.64) NR1H4MRGPRX4LIFR
SCHEMBL2773272 0.85 NR1H4 (0.57) NR1H4
SCHEMBL2770454 0.84 NR1H4 (0.59) NR1H4MRGPRX4VDR
SCHEMBL2773796 0.84 NR1H4 (0.62) NR1H4MRGPRX4LIFR
SCHEMBL2774467 0.83 NR1H4 (0.57) NR1H4
SCHEMBL2772411 0.83 NR1H4 (0.61) NR1H4MRGPRX4LIFR
SCHEMBL2770414 0.83 NR1H4 (0.57) NR1H4MRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029547-B1 FXR AGONISTS LILLY CO ELI (US) 2010-04-28 EP disclosed