SCHEMBL2770441

SCHEMBL2770441

Cc1cc(OCc2c(C(C)C)cnn2-c2c(Cl)cccc2Cl)ccc1N(C)Cc1ccc(C(=O)O)c(C(=O)c2ccccc2)c1

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 17/20 0.54
MRGPRX4 Q96LA9 1/20 0.37
LTC4S Q16873 1/20 0.37
LIFR P42702 1/20 0.35
MCHR1 Q99705 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2770584 0.91 NR1H4 (0.54) NR1H4MRGPRX4MCHR1
SCHEMBL2771344 0.89 NR1H4 (0.51) NR1H4MRGPRX4MCHR1
SCHEMBL2770943 0.89 NR1H4 (0.52) NR1H4MRGPRX4
SCHEMBL2771180 0.89 NR1H4 (0.63) NR1H4MRGPRX4LIFR
SCHEMBL2773103 0.88 NR1H4 (0.52) NR1H4MRGPRX4MCHR1
SCHEMBL2773707 0.88 NR1H4 (0.60) NR1H4MRGPRX4LIFR
SCHEMBL2770617 0.88 NR1H4 (0.51) NR1H4MRGPRX4MCHR1
SCHEMBL2771523 0.88 NR1H4 (0.51) NR1H4
SCHEMBL2770027 0.88 NR1H4 (0.56) NR1H4MCHR1
SCHEMBL2771508 0.87 NR1H4 (0.51) NR1H4MRGPRX4MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029547-B1 FXR AGONISTS LILLY CO ELI (US) 2010-04-28 EP disclosed