SCHEMBL2770587

SCHEMBL2770587

Cc1cc(OCc2c(C(C)C)cnn2-c2c(Cl)cccc2Cl)ccc1C(C)COc1c(C)cccc1C(=O)O

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 12/20 0.55
NPBWR1 P48145 1/20 0.36
MCHR1 Q99705 1/20 0.36
MRGPRX4 Q96LA9 1/20 0.35
NR1I2 O75469 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
BCL2 P10415 2/20 0.33
MCL1 Q07820 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2813670 0.91 NR1H4 (0.57) NR1H4MRGPRX4
SCHEMBL2773667 0.88 NR1H4 (0.56) NR1H4NPBWR1MCHR1MRGPRX4
SCHEMBL2772411 0.88 NR1H4 (0.61) NR1H4MRGPRX4
SCHEMBL2772071 0.88 NR1H4 (0.56) NR1H4MRGPRX4
SCHEMBL2770526 0.87 NR1H4 (0.57) NR1H4NPBWR1MCHR1MRGPRX4
SCHEMBL2771757 0.87 NR1H4 (0.65) NR1H4MRGPRX4
SCHEMBL2770222 0.83 NR1H4 (0.56) NR1H4NPBWR1MCHR1MRGPRX4
SCHEMBL2771111 0.82 NR1H4 (0.58) NR1H4NPBWR1MCHR1MRGPRX4
SCHEMBL2787707 0.82 NR1H4 (0.59) NR1H4MRGPRX4
SCHEMBL2773796 0.80 NR1H4 (0.62) NR1H4MRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029547-B1 FXR AGONISTS LILLY CO ELI (US) 2010-04-28 EP disclosed