SCHEMBL27709592

SCHEMBL27709592

CC(=O)NCc1cc2ncn(-c3cc(C4CC4)[nH]n3)c2cc1NC(C)c1ccc(F)cc1

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 16/20 0.46
MAPK1 P28482 2/20 0.38
JAK2 O60674 1/20 0.38
JAK3 P52333 1/20 0.38
AURKA O14965 1/20 0.36
AURKB Q96GD4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL56702 1.00 NTRK1 (0.46) NTRK1MAPK1JAK2JAK3AURKA
SCHEMBL57581 0.87 NTRK1 (0.49) NTRK1JAK2JAK3AURKAAURKB
SCHEMBL56396 0.84 NTRK1 (0.53) NTRK1JAK2JAK3AURKAAURKB
SCHEMBL57021 0.84 NTRK1 (0.50) NTRK1MAPK1JAK2JAK3AURKA
SCHEMBL56513 0.82 JAK2 (0.52) NTRK1JAK2JAK3AURKAAURKB
SCHEMBL57014 0.79 NTRK1 (0.55) NTRK1JAK2JAK3AURKAAURKB
SCHEMBL57840 0.78 NTRK1 (0.59) NTRK1MAPK1JAK2JAK3AURKA
SCHEMBL57234 0.77 NTRK1 (0.54) NTRK1MAPK1JAK2JAK3AURKA
SCHEMBL4698236 0.76 NTRK1 (0.47) NTRK1JAK2JAK3
SCHEMBL4693863 0.75 NTRK1 (0.44) NTRK1JAK2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101119988-A Chemical compound ASTRAZENECA AB (SE) 2008-02-06 CN claimed
CN-101119988-B Chemical compound ASTRAZENECA AB 2013-03-06 CN disclosed