SCHEMBL27712902

SCHEMBL27712902

CC(=O)N(Cc1ccccc1)n1cccn1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TSPO P30536 1/20 0.40
CRHBP P24387 1/20 0.39
CRHR2 Q13324 1/20 0.39
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
CA12 O43570 1/20 0.39
CA9 Q16790 1/20 0.39
APOBEC3A P31941 2/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
ALOX5 P09917 1/20 0.38
PTGS1 P23219 1/20 0.38
PTGS2 P35354 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30540678 0.89 HTT (0.40) NPC1RAB9ACA12CA9APOBEC3A
SCHEMBL4973158 0.75 CYP19A1 (0.45) ALDH1A1
SCHEMBL27712800 0.73 ELANE (0.37) ALDH1A1LMNA
SCHEMBL16094019 0.72
SCHEMBL11265868 0.70 ELANE (0.34)
SCHEMBL2200339 0.70 NPSR1 (0.38) ALDH1A1LMNA
SCHEMBL9690903 0.70 CHRM2 (0.51) TSPOCRHBPCRHR2NPC1RAB9A
SCHEMBL18429032 0.69 CHRM2 (0.50) TSPOCRHBPCRHR2NPC1RAB9A
SCHEMBL8187887 0.68 KMT2A (0.34) LMNA
SCHEMBL27359652 0.68 KMT2A (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101010315-A Substituted pyrazolyl urea derivatives useful in the treatment of cancer BAYER PHARMACEUTICALS CORP (US) 2007-08-01 CN claimed
CN-101010315-A Substituted pyrazolyl urea derivatives useful in the treatment of cancer BAYER PHARMACEUTICALS CORP (US) 2007-08-01 CN disclosed