SCHEMBL27720455

SCHEMBL27720455

CNc1ccc(NC(=O)c2cc(NC(=O)c3cccc(C(F)(F)F)c3)ccc2C)cn1

nearest known ligand 0.76

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
BRAF P15056 4/20 0.76
CYP2C9 P11712 2/20 0.76
BTK Q06187 11/20 0.75
LCK P06239 10/20 0.75
MAPK14 Q16539 4/20 0.75
KDR P35968 3/20 0.75
KIT P10721 3/20 0.73
CSF1R P07333 2/20 0.72
ABL1 P00519 1/20 0.71
SRC P12931 1/20 0.71
BLK P51451 2/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3929980 0.89 BTK (0.79) BRAFCYP2C9BTKLCKMAPK14
SCHEMBL27720381 0.89 BTK (0.83) BRAFCYP2C9BTKLCKMAPK14
SCHEMBL3939130 0.88 BTK (0.70) BRAFCYP2C9BTKLCKMAPK14
SCHEMBL28768581 0.87 BTK (0.77) BRAFCYP2C9BTKLCKMAPK14
SCHEMBL3929867 0.87 BRAF (1.00) BRAFCYP2C9BTKLCKMAPK14
SCHEMBL2944882 0.86 LCK (1.00) BRAFCYP2C9BTKLCKMAPK14
SCHEMBL3934754 0.85 LCK (0.79) BRAFCYP2C9BTKLCKMAPK14
SCHEMBL2950585 0.84 KDR (1.00) BRAFCYP2C9BTKLCKMAPK14
SCHEMBL1276318 0.84 BRAF (1.00) BRAFBTKLCKMAPK14KDR
SCHEMBL2947918 0.83 LCK (1.00) BRAFCYP2C9BTKLCKMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101128454-A Pyridine carboxamide derivatives for use as anticancer agents ASTRAZENECA AB (SE) 2008-02-20 CN disclosed