SCHEMBL27729014

SCHEMBL27729014

CNCCCOc1cccc2ncnc(Nc3ccc4c(cnn4Cc4ccccn4)c3)c12

nearest known ligand 0.72

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 18/20 0.72
EGFR P00533 4/20 0.68
KCNH2 Q12809 1/20 0.68
ERBB4 Q15303 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4076780 0.98 ERBB2 (0.73) ERBB2EGFRKCNH2ERBB4
SCHEMBL3376303 0.89 ERBB2 (0.77) ERBB2EGFRKCNH2ERBB4
SCHEMBL4080217 0.88 ERBB2 (0.81) ERBB2EGFRKCNH2ERBB4
SCHEMBL4083330 0.87 ERBB2 (0.76) ERBB2EGFRKCNH2ERBB4
SCHEMBL4083320 0.87 ERBB2 (0.76) ERBB2EGFRKCNH2ERBB4
SCHEMBL3376323 0.87 ERBB2 (0.81) ERBB2EGFRKCNH2ERBB4
SCHEMBL27709279 0.86 ERBB2 (0.54) ERBB2EGFRKCNH2ERBB4
SCHEMBL4072543 0.85 ERBB2 (0.71) ERBB2EGFRKCNH2
SCHEMBL3377576 0.85 ERBB2 (0.75) ERBB2EGFRKCNH2ERBB4
SCHEMBL5057307 0.85 ERBB2 (0.78) ERBB2EGFRKCNH2ERBB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101208331-A Quinazoline derivatives as inhibitors of EGF and/or ERBB2 tyrosine kinases ASTRAZENECA AB (SE) 2008-06-25 CN disclosed