SCHEMBL2773167

SCHEMBL2773167

Cc1cc(OCc2c(C(C)C)cnn2-c2c(F)cccc2F)ccc1CNCc1ccc(C(=O)O)cc1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 2/20 0.47
PPARA Q07869 4/20 0.45
SMN1; SMN2 Q16637 1/20 0.42
MAOB P27338 1/20 0.40
KDM4E B2RXH2 1/20 0.38
MRGPRX4 Q96LA9 1/20 0.38
KMT2A Q03164 2/20 0.37
MAPK14 Q16539 1/20 0.36
GCK P35557 1/20 0.36
RXRA P19793 1/20 0.35
RXRB P28702 1/20 0.35
NR4A2 P43354 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2769706 0.93 NR1H4 (0.50) NR1H4PPARASMN1; SMN2MAOBMRGPRX4
SCHEMBL2770618 0.91 NR1H4 (0.58) NR1H4PPARASMN1; SMN2KDM4EMRGPRX4
SCHEMBL2772424 0.85 NR1H4 (0.40) NR1H4PPARASMN1; SMN2MAOBKDM4E
SCHEMBL2773169 0.84 NR1H4 (0.48) NR1H4PPARAMRGPRX4MAPK14RXRA
SCHEMBL2772215 0.84 NR1H4 (0.56) NR1H4PPARAMRGPRX4KMT2A
SCHEMBL2771176 0.84 NR1H4 (0.61) NR1H4PPARASMN1; SMN2MRGPRX4
SCHEMBL2772284 0.84 NR1H4 (0.51) NR1H4MRGPRX4MAPK14RXRARXRB
SCHEMBL2770116 0.84 KDM4E (0.40) NR1H4PPARASMN1; SMN2MAOBKDM4E
SCHEMBL2771059 0.81 NR1H4 (0.57) NR1H4PPARAMAOBMRGPRX4MAPK14
SCHEMBL2771368 0.81 NR1H4 (0.59) NR1H4PPARAMRGPRX4GCKNR4A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029547-B1 FXR AGONISTS LILLY CO ELI (US) 2010-04-28 EP disclosed