SCHEMBL27732136

SCHEMBL27732136

C[C@H](CC(=N)c1ccc2c(C3CCNCC3)ncnc2c1)N(C)C

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAPK7 Q13164 16/20 0.36
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP1A2 P05177 1/20 0.34
HPGD P15428 1/20 0.34
HSD17B10 Q99714 1/20 0.34
KIT P10721 1/20 0.32
SUV39H1 O43463 2/20 0.32
PRMT1 Q99873 2/20 0.32
SMYD3 Q9H7B4 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27711994 0.76 MAPK7 (0.40) MAPK7KITSUV39H1PRMT1SMYD3
SCHEMBL27711985 0.76 MAPK7 (0.40) MAPK7KITSUV39H1PRMT1SMYD3
SCHEMBL5604689 0.75 CYP1A2 (0.42) KDM4EALDH1A1CYP1A2HPGDHSD17B10
SCHEMBL27732137 0.74 MAPK7 (0.37) MAPK7KITSUV39H1PRMT1SMYD3
SCHEMBL21332116 0.71 MAPK7 (0.47) MAPK7KIT
SCHEMBL21332328 0.71 HSP90AB1 (0.41) MAPK7KIT
SCHEMBL27711987 0.69 MAPK7 (0.37) MAPK7KIT
SCHEMBL3570966 0.69 NPC1 (0.47) ALDH1A1CYP1A2KIT
SCHEMBL3563859 0.68 MAPK7 (0.44) MAPK7KIT
SCHEMBL3570195 0.68 MAPK7 (0.53) MAPK7KDM4ECYP1A2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101243065-A Intermediates for the synthesis of alkylquinoline and alkylquinazoline kinase modulators and related synthetic methods JANSSEN PHARMACEUTICA NV (BE) 2008-08-13 CN disclosed