SCHEMBL27733192

SCHEMBL27733192

NCc1cc(Br)ccc1CCCC(=O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F13A1 P00488 3/20 0.43
KDM4E B2RXH2 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
HDAC3 O15379 1/20 0.42
MAPK1 P28482 1/20 0.42
ADRA1A P35348 1/20 0.42
HDAC4 P56524 1/20 0.42
SLC6A3 Q01959 1/20 0.42
HDAC1 Q13547 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC11 Q96DB2 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
HDAC9 Q9UKV0 1/20 0.42
HDAC5 Q9UQL6 1/20 0.42
PTGDR2 Q9Y5Y4 1/20 0.40
MEN1 O00255 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28629668 0.83 F13A1 (0.46) F13A1KDM4ETDP1HDAC3MAPK1
SCHEMBL27491210 0.81 PTGDR2 (0.42) KDM4EPTGDR2MEN1KMT2ALMNA
SCHEMBL19584858 0.80 NPC1 (0.45) F13A1KDM4ETDP1HDAC3MAPK1
SCHEMBL15270886 0.79 POLB (0.49) F13A1KDM4ETDP1HDAC3MAPK1
SCHEMBL3858358 0.78 NPSR1 (0.52) F13A1KDM4ETDP1HDAC3MAPK1
SCHEMBL2818682 0.78 PDPK1 (0.56) F13A1KDM4ETDP1FFAR4
SCHEMBL30917833 0.78 F13A1 (0.44) F13A1KDM4ETDP1HDAC3MAPK1
SCHEMBL28066513 0.77 PTGDR2 (0.42) KDM4EPTGDR2MEN1KMT2ALMNA
SCHEMBL28099899 0.76 KDM4E (0.38) KDM4EPTGDR2
SCHEMBL27812451 0.75 TDP1 (0.37) KDM4ETDP1PTGDR2APEX1GPR17

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101389613-B Macrocyclic factor viia inhibitors useful as anticoagulants BRISTOL MYERS SQUIBB CO 2011-10-12 CN disclosed
CN-101389613-A Macrocyclic factor viia inhibitors useful as anticoagulants BRISTOL MYERS SQUIBB CO (US) 2009-03-18 CN disclosed