SCHEMBL2773377

SCHEMBL2773377

Cc1cc(OCc2c(C(C)C)cnn2-c2c(Cl)cccc2Cl)ccc1-c1ccc2c(C(=O)O)csc2c1

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 17/20 0.52
NR1I2 O75469 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2770660 0.90 NR1H4 (0.49) NR1H4
SCHEMBL2774467 0.88 NR1H4 (0.57) NR1H4
SCHEMBL2773272 0.88 NR1H4 (0.57) NR1H4
SCHEMBL2769974 0.87 NR1H4 (0.48) NR1H4
SCHEMBL2771937 0.87 NR1H4 (0.47) NR1H4CYP1A2CYP2C9
SCHEMBL3150237 0.87 NR1H4 (0.54) NR1H4NR1I2CYP1A2CYP3A4CYP2C9
SCHEMBL2771727 0.86 NR1H4 (0.52) NR1H4
SCHEMBL2771077 0.86 NR1H4 (0.55) NR1H4
SCHEMBL2773254 0.84 NR1H4 (0.52) NR1H4
SCHEMBL2788558 0.84 NR1H4 (0.52) NR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029547-B1 FXR AGONISTS LILLY CO ELI (US) 2010-04-28 EP disclosed