SCHEMBL27739352

SCHEMBL27739352

CC(=O)OC(NC(=O)c1c(C)c(-c2ccccc2)nc2ccccc12)c1ccccn1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 7/20 0.55
CYP3A4 P08684 3/20 0.55
TACR2 P21452 2/20 0.55
TSHR P16473 2/20 0.55
CYP2C9 P11712 2/20 0.55
ALDH1A1 P00352 2/20 0.55
MEN1 O00255 1/20 0.55
TP53 P04637 1/20 0.55
CYP1A2 P05177 1/20 0.55
NFKB1 P19838 1/20 0.55
MAPK1 P28482 1/20 0.55
CYP2C19 P33261 1/20 0.55
BLM P54132 1/20 0.55
PMP22 Q01453 1/20 0.55
KMT2A Q03164 1/20 0.55
ATM Q13315 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
HIF1A Q16665 1/20 0.55
FFAR4 Q5NUL3 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27718254 0.90 TACR3 (0.55) TACR3CYP3A4TACR2CYP2C9CYP1A2
SCHEMBL27739353 0.90 TACR3 (0.55) TACR3TACR2
SCHEMBL28772002 0.85 TACR3 (0.59) TACR3CYP3A4TACR2TSHRCYP2C9
SCHEMBL14094521 0.84 TACR3 (0.60) TACR3CYP3A4TACR2TSHRCYP2C9
SCHEMBL4601948 0.83 TACR3 (0.56) TACR3CYP3A4TACR2TSHRCYP2C9
SCHEMBL27718290 0.82 TACR3 (0.58) TACR3CYP3A4TACR2TSHRCYP2C9
SCHEMBL4602503 0.82 TACR3 (0.75) TACR3CYP3A4TACR2TSHRCYP2C9
SCHEMBL14619204 0.81 TACR3 (0.54) TACR3CYP3A4TACR2TSHRCYP2C9
SCHEMBL27746592 0.77 TACR3 (0.52) TACR3CYP3A4TACR2CYP2C9CYP1A2
SCHEMBL4468216 0.76 TACR3 (0.70) TACR3CYP3A4TACR2TSHRCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101287723-A Amidoalkylpyridylquinolines as NK3 receptor modulators ASTRAZENECA AB (SE) 2008-10-15 CN claimed
CN-101287723-A Amidoalkylpyridylquinolines as NK3 receptor modulators ASTRAZENECA AB (SE) 2008-10-15 CN disclosed