SCHEMBL27740409

SCHEMBL27740409

Cc1ccc(CN(C)CCCCNC(N)=O)cc1C

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
APP P05067 3/20 0.48
TMEM97 Q5BJF2 14/20 0.44
SIGMAR1 Q99720 13/20 0.44
OPRK1 P41145 2/20 0.44
OPRM1 P35372 5/20 0.43
ACKR3 P25106 1/20 0.42
CCR3 P51677 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27719387 0.81 TMEM97 (0.60) APPTMEM97SIGMAR1ACKR3CCR3
SCHEMBL27719409 0.81 APP (0.51) APPTMEM97SIGMAR1OPRK1OPRM1
SCHEMBL4604725 0.77 CHEK1 (0.45) APPTMEM97SIGMAR1OPRM1CCR3
SCHEMBL13989615 0.77 CHRM2 (0.44) SIGMAR1
SCHEMBL4606143 0.73 GSK3A (0.51) CCR3
SCHEMBL14538537 0.73 KMT2A (0.41) APPTMEM97SIGMAR1ACKR3CCR3
SCHEMBL4604262 0.73 LCK (0.48)
SCHEMBL28943830 0.73 CCR3 (0.43) APPTMEM97SIGMAR1OPRK1OPRM1
SCHEMBL18138031 0.70 PARP1 (0.41) SIGMAR1
SCHEMBL7763881 0.69 CHEK1 (0.42) APPTMEM97SIGMAR1ACKR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101296911-A Arylurea derivatives as modulators of chemokine receptor activity NOVARTIS AG (CH) 2008-10-29 CN disclosed