SCHEMBL27748720

SCHEMBL27748720

CC(=O)Oc1ccsc1-n1c(C(C)C)nc2cc(O)ccc2c1=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.50
ESR1 P03372 3/20 0.41
ESR2 Q92731 2/20 0.41
AKR1B1 P15121 1/20 0.35
KDM4E B2RXH2 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
POLB P06746 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
KCNH2 Q12809 1/20 0.31
HRH3 Q9Y5N1 1/20 0.31
PTPN1 P18031 1/20 0.30
PDE10A Q9Y233 1/20 0.30
PKM P14618 1/20 0.30
PARP15 Q460N3 1/20 0.30
PARP10 Q53GL7 1/20 0.30
TNKS2 Q9H2K2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1666166 0.82 TRPV1 (0.51) TRPV1ESR1ESR2AKR1B1KDM4E
SCHEMBL1664223 0.70 TRPV1 (0.55) TRPV1ESR1ESR2KDM4EMAPT
SCHEMBL1664439 0.70 TRPV1 (0.74) TRPV1ESR1ESR2GAAPOLB
SCHEMBL1665294 0.70 TRPV1 (0.70) TRPV1ESR1ESR2AKR1B1GAA
SCHEMBL1663409 0.70 TRPV1 (0.69) TRPV1ESR1ESR2KDM4EMAPT
SCHEMBL1663964 0.70 TRPV1 (0.54) TRPV1ESR1ESR2AKR1B1GAA
SCHEMBL1663637 0.70 TRPV1 (0.65) TRPV1ESR1ESR2AKR1B1KDM4E
SCHEMBL1663398 0.69 TRPV1 (0.72) TRPV1ESR1ESR2KDM4EGAA
SCHEMBL10446158 0.69 TRPV1 (0.72) TRPV1ESR1ESR2KDM4EMAPT
SCHEMBL1664011 0.69 TRPV1 (0.72) TRPV1ESR1ESR2AKR1B1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101356160-A Trisubstituted quinazolinone derivatives as vanilloid antagonists JANSSEN PHARMACEUTICA NV (CH) 2009-01-28 CN disclosed