SCHEMBL27767433

SCHEMBL27767433

NC(=O)c1cc(-c2ccccn2)[nH]c1N(N)C=O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 9/20 0.53
BTK Q06187 1/20 0.41
JAK2 O60674 3/20 0.40
CCNB2 O95067 2/20 0.40
CDK1 P06493 2/20 0.40
CCNB1 P14635 2/20 0.40
GSK3B P49841 2/20 0.40
CCNB3 Q8WWL7 2/20 0.40
CCNA2 P20248 2/20 0.40
CDK2 P24941 2/20 0.40
CCNA1 P78396 2/20 0.40
IKBKB O14920 1/20 0.40
CCNT1 O60563 1/20 0.40
CCNE2 O96020 1/20 0.40
PRKCB P05771 1/20 0.40
CCNE1 P24864 1/20 0.40
CDK9 P50750 1/20 0.40
TAOK1 Q7L7X3 1/20 0.40
PARP1 P09874 1/20 0.40
DHODH Q02127 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27788862 0.80 BRD4 (0.56) CDC7JAK2CCNB2CDK1CCNB1
SCHEMBL27789086 0.78 BRD4 (0.44) CDC7CCNB2CDK1CCNB1GSK3B
SCHEMBL4342616 0.77 CDC7 (0.61) CDC7BTKJAK2CCNB2CDK1
SCHEMBL27767422 0.76 CDC7 (0.47) CDC7BTKPARP1NPC1RAB9A
SCHEMBL27767424 0.76 IKBKB (0.43) CDC7JAK2IKBKBPARP1KDM4E
SCHEMBL27788867 0.74 BRD4 (0.40) CDC7CCNA2CDK2CCNA1PARP1
SCHEMBL27788861 0.74 BRD4 (0.41) CDC7CCNA2CDK2CCNA1PARP1
SCHEMBL2198743 0.74 CDC7 (0.54) CDC7BTKJAK2CCNB2CDK1
SCHEMBL27767442 0.73 PARP1 (0.43) CDC7CCNA2CDK2CCNA1PARP1
SCHEMBL27767426 0.73 CDC7 (0.43) CDC7BTKCCNB2CDK1CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101622229-B Pyrrole derivatives having ureido and aminocarbonyl groups as substituents SANTEN PHARMACEUTICAL CO LTD 2013-02-27 CN claimed
CN-101622229-A Novel pyrrole derivatives having ureido group and aminocarbonyl group as substituents SANTEN PHARMACEUTICAL CO LTD 2010-01-06 CN claimed
CN-101622229-B Pyrrole derivatives having ureido and aminocarbonyl groups as substituents SANTEN PHARMACEUTICAL CO LTD 2013-02-27 CN disclosed
CN-101622229-A Novel pyrrole derivatives having ureido group and aminocarbonyl group as substituents SANTEN PHARMACEUTICAL CO LTD 2010-01-06 CN disclosed