SCHEMBL27768315

SCHEMBL27768315

CN(C=O)c1nnc(CC2CCNC2)c2cc(-c3ccc(Cl)cc3)sc12

nearest known ligand 0.41

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 17/20 0.41
MCHR1 Q99705 2/20 0.36
KCNH2 Q12809 2/20 0.35
CDK2AP1 O14519 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23630273 0.95 CHEK1 (0.46) CHEK1KCNH2CDK2AP1
SCHEMBL28781348 0.84 MCHR1 (0.39) CHEK1MCHR1
SCHEMBL8835231 0.83 CHEK1 (0.49) CHEK1MCHR1KCNH2CDK2AP1
SCHEMBL26983380 0.82 MCHR1 (0.35) CHEK1MCHR1KCNH2
SCHEMBL27768305 0.81 CHEK1 (0.62) CHEK1CDK2AP1
SCHEMBL8831254 0.81 CHEK1 (0.62) CHEK1CDK2AP1
Hydrochloric Acid SCHEMBL27768311 0.80 CHEK1 (0.61) CHEK1CDK2AP1
SCHEMBL29012208 0.79 CHEK1 (0.49) CHEK1MCHR1CDK2AP1
SCHEMBL8832033 0.79 CHEK1 (0.51) CHEK1MCHR1CDK2AP1
SCHEMBL8835672 0.78 CHEK1 (0.54) CHEK1KCNH2CDK2AP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101481380-A Thiofuran pyridazine compound, preparation thereof, pharmaceutical composition and uses thereof ZHEJIANG MEDICINE CO LTD (CN) 2009-07-15 CN claimed
CN-101481380-A Thiofuran pyridazine compound, preparation thereof, pharmaceutical composition and uses thereof ZHEJIANG MEDICINE CO LTD (CN) 2009-07-15 CN disclosed