SCHEMBL27768321

SCHEMBL27768321

O=C(OF)C(O)(c1ccccc1)c1ccc(F)c(F)c1F

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.38
KCNN4 O15554 6/20 0.36
ALDH1A1 P00352 2/20 0.35
HTT P42858 1/20 0.35
MCOLN3 Q8TDD5 1/20 0.35
CHRM3 P20309 3/20 0.34
CHRM2 P08172 2/20 0.34
CHRM1 P11229 2/20 0.34
MEN1 O00255 1/20 0.34
POLB P06746 1/20 0.34
KMT2A Q03164 1/20 0.34
CHRM4 P08173 1/20 0.33
KCNE1 P15382 1/20 0.33
KCNQ1 P51787 1/20 0.33
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27789581 0.83 KCNN4 (0.50) CYP2C9KCNN4ALDH1A1HTTMCOLN3
SCHEMBL28049560 0.80 CHRM3 (0.46) CYP2C9KCNN4ALDH1A1CHRM3CHRM2
SCHEMBL4160700 0.74 KCNN4 (0.37) CYP2C9KCNN4ALDH1A1HTTMCOLN3
SCHEMBL29101509 0.73 CYP3A4 (0.41) CYP2C9KCNN4ALDH1A1KCNE1KCNQ1
SCHEMBL3818507 0.71 CYP2C9 (0.50) CYP2C9KCNN4ALDH1A1HTTMCOLN3
SCHEMBL28743258 0.71 POLB (0.44) ALDH1A1HTTCHRM3CHRM2CHRM1
SCHEMBL4160698 0.70 CYP2C9 (0.49) CYP2C9KCNN4ALDH1A1HTTMCOLN3
SCHEMBL30097456 0.70 CES1 (0.38) KCNN4ALDH1A1HTTMCOLN3POLB
Bromomethane SCHEMBL3192554 0.68 CYP2C9 (0.46) CYP2C9KCNN4ALDH1A1HTTMCOLN3
SCHEMBL28381845 0.68 KCNN4 (0.41) KCNN4ALDH1A1KCNE1KCNQ1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103497185-A Pyrazolo(3, 4-B)pyridine derivatives as phosphodiesterase inhibitors RANBAXY LAB LTD 2014-01-08 CN disclosed
CN-102256963-A Cyclic pyrimidine-4-carboxamides as CCR2 receptor antagonists for the treatment of inflammation, asthma and COPD BOEHRINGER INGELHEIM INT 2011-11-23 CN disclosed
CN-101980742-A Inhaler VECTURA DELIVERY DEVICES LTD (GB) 2011-02-23 CN disclosed
CN-101801376-A Pyrazolo (3,4-b) pyridine derivatives as phosphodiesterase inhibitors RANBAXY LAB LTD 2010-08-11 CN disclosed
CN-101616901-A Inhibitors of phosphodiesterase type IV RANBAXY LAB LTD 2009-12-30 CN disclosed