SCHEMBL27771679

SCHEMBL27771679

Cc1nc2c(c(-c3ccccc3Cl)c1CN)C(=O)N([C@@H](OC(=O)C(F)(F)F)C(=O)N(C)C)CC2

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 20/20 0.46
DPP8 Q6V1X1 16/20 0.36
DPP9 Q86TI2 15/20 0.36
CYP3A4 P08684 5/20 0.34
CYP2C19 P33261 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27771680 1.00 DPP4 (0.46) DPP4DPP8DPP9CYP3A4CYP2C19
SCHEMBL294870 0.76 DPP4 (0.54) DPP4DPP8DPP9CYP3A4CYP2C19
SCHEMBL294679 0.66 DPP4 (0.68) DPP4DPP8DPP9CYP3A4CYP2C19
SCHEMBL295145 0.64 DPP4 (0.75) DPP4DPP8DPP9CYP3A4CYP2C19
SCHEMBL294346 0.64 DPP4 (1.00) DPP4DPP8DPP9CYP3A4CYP2C19
SCHEMBL294237 0.63 DPP4 (0.67) DPP4DPP8DPP9CYP3A4CYP2C19
SCHEMBL4404901 0.62 DPP4 (0.43) DPP4DPP8DPP9CYP3A4CYP2C19
SCHEMBL2703689 0.62 DPP4 (0.57) DPP4DPP8DPP9CYP3A4CYP2C19
SCHEMBL2703685 0.62 DPP4 (0.57) DPP4DPP8DPP9CYP3A4CYP2C19
SCHEMBL294677 0.62 DPP4 (0.69) DPP4DPP8DPP9CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101595109-A 7, 8-dihydro-1, 6-naphthyridin-5 (6H) -ones and related bicyclic compounds as dipeptidyl peptidase IV inhibitors and methods BRISTOL MYERS SQUIBB CO (US) 2009-12-02 CN disclosed