SCHEMBL27782820

SCHEMBL27782820

Cc1cc(C(=O)c2c[nH]c3ncc(-c4cccc(C(=O)N=[N+]=[N-])c4)cc23)nn1C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 2/20 0.44
AXL P30530 5/20 0.42
PAK1 Q13153 5/20 0.41
NEK1 Q96PY6 5/20 0.41
CYP3A4 P08684 1/20 0.40
MAP4K1 Q92918 1/20 0.40
CDC7 O00311 1/20 0.40
PLK4 O00444 1/20 0.40
CHEK1 O14757 1/20 0.40
AURKA O14965 1/20 0.40
MAPK13 O15264 1/20 0.40
PDPK1 O15530 1/20 0.40
DYRK3 O43781 1/20 0.40
ROCK2 O75116 1/20 0.40
RPS6KA5 O75582 1/20 0.40
PRKD3 O94806 1/20 0.40
PAK4 O96013 1/20 0.40
CHEK2 O96017 1/20 0.40
ABL1 P00519 1/20 0.40
EGFR P00533 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27804369 0.91 AAK1 (0.42) AAK1AXLPAK1BRD4PKN1
SCHEMBL10263401 0.86 AAK1 (0.49) AAK1AXLPAK1NEK1CYP3A4
SCHEMBL27782909 0.86 AAK1 (0.44) AAK1AXLPAK1NEK1CYP3A4
SCHEMBL858062 0.86 AXL (0.56) AAK1AXLPAK1NEK1CYP3A4
SCHEMBL857911 0.83 KIT (0.52) AAK1AXLPAK1NTRK1DYRK1A
SCHEMBL858780 0.80 BRD4 (0.51) AAK1AXLPAK1NEK1NTRK1
SCHEMBL4301666 0.79 PIK3CA (0.51) AXLPAK1NTRK1ITKDYRK1A
SCHEMBL859107 0.78 AXL (0.45) AAK1AXLPAK1NEK1CDC7
SCHEMBL1364902 0.78 AXL (0.45) AAK1AXLPAK1NEK1CDC7
SCHEMBL857852 0.78 MAP3K11 (0.49) AAK1AXLPAK1CDC7PLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1925855-B Compounds and methods for development of Ret modulators PLEXXIKON INC 2010-06-16 CN claimed