SCHEMBL27782831

SCHEMBL27782831

FC(F)(F)c1ccc2ncncc2c1

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EGFR P00533 9/20 0.55
BACE1 P56817 1/20 0.47
PIK3CD O00329 1/20 0.46
PIK3CA P42336 1/20 0.46
KDM4E B2RXH2 1/20 0.43
EPHX2 P34913 1/20 0.41
SCN4A P35499 1/20 0.41
FGFR4 P22455 1/20 0.40
METAP2 P50579 1/20 0.40
TDO2 P48775 1/20 0.39
AR P10275 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30056467 1.00 EGFR (0.55) EGFRBACE1PIK3CDPIK3CAKDM4E
SCHEMBL28128190 0.85 EGFR (0.55) EGFRBACE1KDM4EMETAP2TDO2
SCHEMBL31139918 0.82 BACE1 (0.45) EGFRBACE1KDM4EEPHX2SCN4A
SCHEMBL10280767 0.81 EGFR (0.55) EGFRPIK3CDPIK3CAFGFR4METAP2
SCHEMBL20132505 0.79 EGFR (0.51) EGFRPIK3CDPIK3CAFGFR4TDO2
SCHEMBL17410801 0.75 EGFR (0.60) EGFRBACE1PIK3CDPIK3CAKDM4E
SCHEMBL29891394 0.75 EGFR (0.60) EGFRBACE1PIK3CDPIK3CAKDM4E
SCHEMBL7155460 0.74 NPC1 (0.44) EGFR
SCHEMBL8644295 0.74 PIK3CA (0.73) EGFRPIK3CDPIK3CAKDM4EFGFR4
SCHEMBL25228140 0.74 EGFR (0.54) EGFRPIK3CDPIK3CAFGFR4TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101568532-A Cyclic derivatives as modulators of chemokine receptor activity BRISTOL MYERS SQUIBB CO (US) 2009-10-28 CN disclosed