SCHEMBL27785877

SCHEMBL27785877

FC(F)(F)Nc1nnc(-c2ncccc2OCc2ccncc2)o1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDR P35968 15/20 0.41
FLT1 P17948 14/20 0.41
CDC7 O00311 1/20 0.38
CCNE1 P24864 1/20 0.38
CDK2 P24941 1/20 0.38
DBF4 Q9UBU7 1/20 0.38
ALDH1A1 P00352 2/20 0.37
LMNA P02545 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
KDM4E B2RXH2 1/20 0.36
USP2 O75604 1/20 0.36
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36
ABCB1 P08183 1/20 0.36
MEN1 O00255 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1347109 0.82 KDR (0.52) KDRFLT1ALDH1A1LMNASMN1; SMN2
SCHEMBL1346532 0.68 KDR (0.56) KDRFLT1KDM4ERAB9A
SCHEMBL1346273 0.65 KDR (0.66) KDRFLT1
SCHEMBL1346648 0.65 KDR (0.53) KDRFLT1
SCHEMBL6026657 0.63 NPC1 (0.74) ALDH1A1LMNASMN1; SMN2KDM4EHSD17B10
SCHEMBL2385077 0.63 ABCB1 (0.51) ALDH1A1LMNASMN1; SMN2ABCB1MEN1
SCHEMBL30887571 0.63 ABCB1 (0.51) ALDH1A1LMNASMN1; SMN2ABCB1MEN1
SCHEMBL1346514 0.62 KDR (0.45) KDRFLT1ALDH1A1LMNASMN1; SMN2
SCHEMBL27764283 0.60 KDM4E (0.45) KDRFLT1ALDH1A1LMNASMN1; SMN2
SCHEMBL25389540 0.59 NPC1 (0.49) ALDH1A1LMNASMN1; SMN2KDM4EUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101600712-A Novel oxadiazole derivative and thiadiazole derivative having angiogenesis inhibitory activity SANTEN PHARMACEUTICAL CO LTD (JP) 2009-12-09 CN claimed
CN-103224493-A Novel oxadiazole derivatives and thiadiazole derivatives having neovascularization inhibitory activity SANTEN PHARMACEUTICAL CO LTD 2013-07-31 CN disclosed
CN-101600712-A Novel oxadiazole derivative and thiadiazole derivative having angiogenesis inhibitory activity SANTEN PHARMACEUTICAL CO LTD (JP) 2009-12-09 CN disclosed