SCHEMBL27787161

SCHEMBL27787161

CC(C=O)c1ccc(NCc2ccc(C(F)(F)F)cc2)nc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 2/20 0.47
KIT P10721 1/20 0.47
RAB9A P51151 3/20 0.46
MAPT P10636 3/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
NPC1 O15118 2/20 0.46
ALDH1A1 P00352 2/20 0.46
GAA P10253 2/20 0.44
LMNA P02545 1/20 0.44
HTT P42858 1/20 0.44
VNN1 O95497 2/20 0.43
HDAC3 O15379 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
EPHX2 P34913 1/20 0.42
ASPH Q12797 2/20 0.40
KDM8 Q8N371 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27787159 0.84 HDAC3 (0.49) CSF1RKITRAB9AMAPTMEN1
SCHEMBL3813790 0.79 CSF1R (0.52) CSF1RKITRAB9AMAPTMEN1
SCHEMBL1267411 0.79 CSF1R (0.49) CSF1RKITRAB9AMAPTMEN1
SCHEMBL1508500 0.74 FFAR1 (0.62) CSF1RHDAC3HDAC1HDAC2HDAC6
SCHEMBL1508369 0.74 CSF1R (0.44) CSF1RKITRAB9AMAPTMEN1
SCHEMBL1267867 0.73 HDAC3 (0.57) CSF1RKITRAB9AMAPTMEN1
SCHEMBL1266913 0.73 NPC1 (0.58) CSF1RKITRAB9AMAPTMEN1
SCHEMBL2702140 0.73 PDE2A (0.46)
SCHEMBL23260548 0.73 LSS (0.51) CSF1RKITRAB9AMAPTMEN1
SCHEMBL28780861 0.72 NPC1 (0.57) CSF1RKITRAB9AMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103497188-A Compounds modulating c-fms and/or c-kit activity and uses therefor PLEXXIKON INC 2014-01-08 CN disclosed
CN-101605787-B Compounds that modulate c-fms and/or c-kit activity and uses thereof PLEXXIKON INC 2013-11-13 CN disclosed
CN-101605787-A Compounds that modulate c-fms and/or c-kit activity and uses thereof PLEXXIKON INC (US) 2009-12-16 CN disclosed