SCHEMBL27788313

SCHEMBL27788313

SC(c1nnc(-c2cccc(Cl)c2)o1)c1nnc(-c2ccncc2)n1C1CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.52
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
TP53 P04637 2/20 0.39
TSHR P16473 1/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
PIM1 P11309 1/20 0.39
BCHE P06276 1/20 0.38
CYP3A4 P08684 1/20 0.38
POLB P06746 1/20 0.37
NOTUM Q6P988 1/20 0.36
GSK3B P49841 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
CALCRL Q16602 1/20 0.35
MAPT P10636 2/20 0.35
CA1 P00915 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4331659 0.86 KCNH2 (0.54) KCNH2NPC1RAB9ATP53TSHR
SCHEMBL1544228 0.85 KCNH2 (0.39) KCNH2NPC1RAB9ATP53TSHR
SCHEMBL27788275 0.85 BCHE (0.37) KCNH2NPC1RAB9ATP53SMN1; SMN2
SCHEMBL27788283 0.85 KCNH2 (0.41) KCNH2NPC1RAB9ABCHECYP3A4
SCHEMBL1543777 0.84 TLR8 (0.40) KCNH2CYP3A4MEN1KMT2A
SCHEMBL27810138 0.84 KCNH2 (0.66) KCNH2NPC1RAB9ATP53TSHR
SCHEMBL27788491 0.83 KCNH2 (0.54) KCNH2NPC1RAB9ATP53TSHR
SCHEMBL1543853 0.82 KCNH2 (0.54) KCNH2NPC1RAB9ATP53TSHR
SCHEMBL1543735 0.82 KCNH2 (0.54) KCNH2NPC1RAB9ATP53TSHR
SCHEMBL1544379 0.82 KCNH2 (0.54) KCNH2NPC1RAB9ATP53TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101723941-A “1,2,4” oxadiazole as a metabotropic glutamate receptor-5 modulator ASTRAZENECA AB 2010-06-09 CN claimed
CN-101723941-A “1,2,4” oxadiazole as a metabotropic glutamate receptor-5 modulator ASTRAZENECA AB 2010-06-09 CN disclosed