SCHEMBL2779675

SCHEMBL2779675

COC(=O)c1c[nH]c2ccc(C3(Cc4cccc(OC)c4)CC(=O)N(Cc4ccccc4)C3=O)cc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 2/20 0.46
GABRP O00591 3/20 0.46
GABRD O14764 3/20 0.46
GABRA1 P14867 3/20 0.46
GABRB1 P18505 3/20 0.46
GABRG2 P18507 3/20 0.46
GABRB3 P28472 3/20 0.46
GABRA5 P31644 3/20 0.46
GABRA3 P34903 3/20 0.46
GABRA2 P47869 3/20 0.46
GABRB2 P47870 3/20 0.46
GABRA4 P48169 3/20 0.46
GABRE P78334 3/20 0.46
GABRA6 Q16445 3/20 0.46
GABRG1 Q8N1C3 3/20 0.46
GABRG3 Q99928 3/20 0.46
GABRQ Q9UN88 3/20 0.46
ACHE P22303 1/20 0.43
PTGDR2 Q9Y5Y4 4/20 0.42
HAT1 O14929 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2778430 0.88 NR4A2 (0.43) NR4A2GABRPGABRDGABRA1GABRB1
SCHEMBL2779691 0.86 NR4A2 (0.45) NR4A2GABRPGABRDGABRA1GABRB1
SCHEMBL2781901 0.85 NR4A2 (0.41) NR4A2GABRPGABRDGABRA1GABRB1
SCHEMBL2780123 0.85 NR4A2 (0.44) NR4A2GABRPGABRDGABRA1GABRB1
SCHEMBL2780111 0.82 NR4A2 (0.48) NR4A2GABRPGABRDGABRA1GABRB1
SCHEMBL985058 0.81 SLC6A2 (0.53) PTGDR2NR3C2SIGMAR1
SCHEMBL983940 0.76 PTGDR2 (0.43) PTGDR2NR3C2
SCHEMBL2778867 0.71 NR4A2 (0.49) NR4A2GABRA1GABRB1GABRA3GABRB2
SCHEMBL2777419 0.69 NR4A2 (0.49) NR4A2ACHE
SCHEMBL984732 0.69 SLC6A2 (0.48) ACHEPTGDR2SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257545-A1 PYRROLIDINYL DERIVATIVES AND USES THEREOF F. Hoffmann-La Roche AG (CH) 2010-12-08 EP disclosed
WO-2009115427-A1 PYRROLIDINYL DERIVATIVES AND USES THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2009-09-24 WO disclosed