SCHEMBL27797643

SCHEMBL27797643

Cc1cc(C23CC4CC(CC(C4)C2)C3)c(O)cc1N=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 3/20 0.41
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
THRB P10828 1/20 0.40
RECQL P46063 1/20 0.40
NR2E1 Q9Y466 1/20 0.40
RARA P10276 6/20 0.39
RARB P10826 4/20 0.39
RARG P13631 4/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
TP53 P04637 1/20 0.39
CYP3A4 P08684 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
ALOX15 P16050 1/20 0.39
ALOX12 P18054 1/20 0.39
MAPK1 P28482 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL549772 0.80 MEN1 (0.44) IKBKBMEN1KMT2ATHRBRECQL
SCHEMBL549599 0.77 IKBKB (0.45) IKBKBMEN1KMT2ATHRBRECQL
SCHEMBL436182 0.76 MEN1 (0.41) IKBKBMEN1KMT2ATHRBRECQL
SCHEMBL548836 0.76 MEN1 (0.53) IKBKBMEN1KMT2ATHRBRECQL
SCHEMBL548705 0.75 MEN1 (0.46) IKBKBMEN1KMT2ATHRBRECQL
SCHEMBL548700 0.74 MEN1 (0.52) IKBKBMEN1KMT2ATHRBRECQL
SCHEMBL27448235 0.74 MEN1 (0.44) IKBKBMEN1KMT2ATHRBRECQL
SCHEMBL436214 0.74 IKBKB (0.39) IKBKBMEN1KMT2ATHRBRECQL
SCHEMBL1914338 0.73 IKBKB (0.43) IKBKBMEN1KMT2ATHRBRECQL
SCHEMBL549542 0.73 MEN1 (0.50) IKBKBMEN1KMT2ATHRBRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107501099-A The adjusting control agent of ATP combination cassette transporters 沃泰克斯药物股份有限公司 2017-12-22 CN disclosed
CN-104788328-B The adjusting control agent of ATP combination cassette transporters 沃泰克斯药物股份有限公司 2017-09-12 CN disclosed
CN-101935301-A Modulators of ATP-binding cassette transporters VERTEX PHARMA 2011-01-05 CN disclosed
CN-101891680-A The adjusting control agent of ATP- combination cassette transporters VERTEX PHARMA 2010-11-24 CN disclosed