SCHEMBL27798142

SCHEMBL27798142

O=C1NC(=O)c2cc([N+](=O)[O-])ccc21.[KH]

nearest known ligand 0.96

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.96
TDP1 Q9NUW8 1/20 0.96
PTPRC P08575 3/20 0.60
S100A4 P26447 2/20 0.60
ALDH1A1 P00352 3/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
CASP3 P42574 3/20 0.59
CAPN9 O14815 1/20 0.59
MEN1 O00255 3/20 0.58
KMT2A Q03164 3/20 0.58
TDP2 O95551 1/20 0.58
MAPT P10636 3/20 0.56
CA9 Q16790 2/20 0.56
CA1 P00915 1/20 0.56
CA2 P00918 1/20 0.56
CA7 P43166 1/20 0.56
BCHE P06276 1/20 0.53
ACHE P22303 1/20 0.53
CES1 P23141 1/20 0.53
KDM4E B2RXH2 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL151957 0.98 CYP3A4 (1.00) CYP3A4TDP1PTPRCS100A4ALDH1A1
Methane SCHEMBL28326322 0.96 CYP3A4 (0.96) CYP3A4TDP1PTPRCS100A4ALDH1A1
SCHEMBL3134182 0.84 TDP1 (0.74) CYP3A4TDP1PTPRCS100A4ALDH1A1
SCHEMBL29202832 0.83 CYP3A4 (0.71) CYP3A4TDP1PTPRCS100A4ALDH1A1
SCHEMBL27559675 0.83 CYP3A4 (0.71) CYP3A4TDP1PTPRCS100A4ALDH1A1
SCHEMBL177892 0.80 CYP3A4 (0.68) CYP3A4TDP1ALDH1A1SMN1; SMN2CASP3
Phthalimide SCHEMBL27559674 0.80 CYP3A4 (0.67) CYP3A4TDP1PTPRCS100A4ALDH1A1
SCHEMBL3566821 0.78 CYP3A4 (0.65) CYP3A4TDP1PTPRCS100A4ALDH1A1
SCHEMBL3566817 0.78 CYP3A4 (0.65) CYP3A4TDP1PTPRCS100A4ALDH1A1
SCHEMBL16303093 0.78 CYP3A4 (0.67) CYP3A4TDP1ALDH1A1SMN1; SMN2CASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101898985-B N-substituted benzenesulfonyl-substituted benzamides small molecular inhibitor of Bcl-2 protein and application thereof UNIV PLA 2ND MILITARY MEDICAL 2014-05-28 CN disclosed
CN-101899008-B N-substituted pyrimidine sulfonyl-substituted benzamide type small molecular inhibitor for Bcl-2 protein and application thereof UNIV PLA 2ND MILITARY MEDICAL 2012-10-17 CN disclosed
CN-101899008-A N-substituted pyrimidine sulfonyl-substituted benzamide type small molecular inhibitor for Bcl-2 protein and application thereof UNIV PLA 2ND MILITARY MEDICAL 2010-12-01 CN disclosed
CN-101898985-A N-substituted benzenesulfonyl-substituted benzamides small molecular inhibitor of Bcl-2 protein and application thereof UNIV PLA 2ND MILITARY MEDICAL 2010-12-01 CN disclosed